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Effect of mofezolac-galactose distance in conjugates targeting cyclooxygenase (COX)-1 and CNS GLUT-1 carrier.
Perrone, Maria Grazia; Vitale, Paola; Ferorelli, Savina; Boccarelli, Angelina; Coluccia, Mauro; Pannunzio, Alessandra; Campanella, Federica; Di Mauro, Giuseppe; Bonaccorso, Carmela; Fortuna, Cosimo G; Scilimati, Antonio.
Afiliação
  • Perrone MG; Department of Pharmacy - Pharmaceutical Sciences, University of Bari "Aldo Moro", Via E. Orabona 4, 70125 Bari, Italy.
  • Vitale P; Department of Pharmacy - Pharmaceutical Sciences, University of Bari "Aldo Moro", Via E. Orabona 4, 70125 Bari, Italy.
  • Ferorelli S; Department of Pharmacy - Pharmaceutical Sciences, University of Bari "Aldo Moro", Via E. Orabona 4, 70125 Bari, Italy.
  • Boccarelli A; Department of Biomedical Sciences and Human Oncology, University of Bari "Aldo Moro", Piazza Giulio Cesare 11, 70124 Bari, Italy.
  • Coluccia M; Department of Pharmacy - Pharmaceutical Sciences, University of Bari "Aldo Moro", Via E. Orabona 4, 70125 Bari, Italy.
  • Pannunzio A; Department of Pharmacy - Pharmaceutical Sciences, University of Bari "Aldo Moro", Via E. Orabona 4, 70125 Bari, Italy.
  • Campanella F; Department of Pharmacy - Pharmaceutical Sciences, University of Bari "Aldo Moro", Via E. Orabona 4, 70125 Bari, Italy.
  • Di Mauro G; Department of Chemical Science, University of Catania, Viale Andrea Doria 6, 95125 Catania, Italy.
  • Bonaccorso C; Department of Chemical Science, University of Catania, Viale Andrea Doria 6, 95125 Catania, Italy.
  • Fortuna CG; Department of Chemical Science, University of Catania, Viale Andrea Doria 6, 95125 Catania, Italy.
  • Scilimati A; Department of Pharmacy - Pharmaceutical Sciences, University of Bari "Aldo Moro", Via E. Orabona 4, 70125 Bari, Italy. Electronic address: antonio.scilimati@uniba.it.
Eur J Med Chem ; 141: 404-416, 2017 Dec 01.
Article em En | MEDLINE | ID: mdl-29032033

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Sistema Nervoso Central / Inibidores de Ciclo-Oxigenase / Ciclo-Oxigenase 1 / Transportador de Glucose Tipo 1 / Galactose / Isoxazóis Limite: Animals / Humans Idioma: En Ano de publicação: 2017 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Sistema Nervoso Central / Inibidores de Ciclo-Oxigenase / Ciclo-Oxigenase 1 / Transportador de Glucose Tipo 1 / Galactose / Isoxazóis Limite: Animals / Humans Idioma: En Ano de publicação: 2017 Tipo de documento: Article