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Identification of novel leishmanicidal molecules by virtual and biochemical screenings targeting Leishmania eukaryotic translation initiation factor 4A.
Harigua-Souiai, Emna; Abdelkrim, Yosser Zina; Bassoumi-Jamoussi, Imen; Zakraoui, Ons; Bouvier, Guillaume; Essafi-Benkhadir, Khadija; Banroques, Josette; Desdouits, Nathan; Munier-Lehmann, Hélène; Barhoumi, Mourad; Tanner, N Kyle; Nilges, Michael; Blondel, Arnaud; Guizani, Ikram.
Afiliação
  • Harigua-Souiai E; Laboratory of Molecular Epidemiology and Experimental Pathology - LR11IPT04, Institut Pasteur de Tunis, Université de Tunis el Manar, Tunis, Tunisia.
  • Abdelkrim YZ; Institut Pasteur, Unité de Bioinformatique Structurale, CNRS UMR 3528, Département de Biologie Structurale et Chimie, Paris, France.
  • Bassoumi-Jamoussi I; Laboratory of Molecular Epidemiology and Experimental Pathology - LR11IPT04, Institut Pasteur de Tunis, Université de Tunis el Manar, Tunis, Tunisia.
  • Zakraoui O; Laboratory of Microbial Gene Expression (EGM), CNRS UMR8261/Université Paris Diderot P7, Sorbonne Paris Cité & PSL, Institut de Biologie Physico-Chimique, Paris, France.
  • Bouvier G; Faculté des Sciences de Bizerte, Université de Carthage, Tunis, Tunisia.
  • Essafi-Benkhadir K; Laboratory of Molecular Epidemiology and Experimental Pathology - LR11IPT04, Institut Pasteur de Tunis, Université de Tunis el Manar, Tunis, Tunisia.
  • Banroques J; Laboratory of Molecular Epidemiology and Experimental Pathology - LR11IPT04, Institut Pasteur de Tunis, Université de Tunis el Manar, Tunis, Tunisia.
  • Desdouits N; Institut Pasteur, Unité de Bioinformatique Structurale, CNRS UMR 3528, Département de Biologie Structurale et Chimie, Paris, France.
  • Munier-Lehmann H; Laboratory of Molecular Epidemiology and Experimental Pathology - LR11IPT04, Institut Pasteur de Tunis, Université de Tunis el Manar, Tunis, Tunisia.
  • Barhoumi M; Laboratory of Microbial Gene Expression (EGM), CNRS UMR8261/Université Paris Diderot P7, Sorbonne Paris Cité & PSL, Institut de Biologie Physico-Chimique, Paris, France.
  • Tanner NK; Institut Pasteur, Unité de Bioinformatique Structurale, CNRS UMR 3528, Département de Biologie Structurale et Chimie, Paris, France.
  • Nilges M; Institut Pasteur, Unité de Chimie et Biocatalyse, Département de Biologie Structurale et Chimie, Paris, France.
  • Blondel A; Unité Mixte de Recherche 3523, Centre National de la Recherche Scientifique, Paris, France.
  • Guizani I; Laboratory of Molecular Epidemiology and Experimental Pathology - LR11IPT04, Institut Pasteur de Tunis, Université de Tunis el Manar, Tunis, Tunisia.
PLoS Negl Trop Dis ; 12(1): e0006160, 2018 01.
Article em En | MEDLINE | ID: mdl-29346371

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Leishmania infantum / Fator de Iniciação 4A em Eucariotos / Avaliação Pré-Clínica de Medicamentos / Antiprotozoários Tipo de estudo: Diagnostic_studies / Prognostic_studies Idioma: En Ano de publicação: 2018 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Leishmania infantum / Fator de Iniciação 4A em Eucariotos / Avaliação Pré-Clínica de Medicamentos / Antiprotozoários Tipo de estudo: Diagnostic_studies / Prognostic_studies Idioma: En Ano de publicação: 2018 Tipo de documento: Article