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Treatment with HC-070, a potent inhibitor of TRPC4 and TRPC5, leads to anxiolytic and antidepressant effects in mice.
Just, Stefan; Chenard, Bertrand L; Ceci, Angelo; Strassmaier, Timothy; Chong, Jayhong A; Blair, Nathaniel T; Gallaschun, Randall J; Del Camino, Donato; Cantin, Susan; D'Amours, Marc; Eickmeier, Christian; Fanger, Christopher M; Hecker, Carsten; Hessler, David P; Hengerer, Bastian; Kroker, Katja S; Malekiani, Sam; Mihalek, Robert; McLaughlin, Joseph; Rast, Georg; Witek, JoAnn; Sauer, Achim; Pryce, Christopher R; Moran, Magdalene M.
Afiliação
  • Just S; Boehringer Ingelheim Pharma GmbH & Co. KG, Biberach an der Riss, Germany.
  • Chenard BL; Hydra Biosciences, Cambridge, Massachusetts, United States of America.
  • Ceci A; Boehringer Ingelheim Pharma GmbH & Co. KG, Biberach an der Riss, Germany.
  • Strassmaier T; Hydra Biosciences, Cambridge, Massachusetts, United States of America.
  • Chong JA; Hydra Biosciences, Cambridge, Massachusetts, United States of America.
  • Blair NT; Hydra Biosciences, Cambridge, Massachusetts, United States of America.
  • Gallaschun RJ; Hydra Biosciences, Cambridge, Massachusetts, United States of America.
  • Del Camino D; Hydra Biosciences, Cambridge, Massachusetts, United States of America.
  • Cantin S; Hydra Biosciences, Cambridge, Massachusetts, United States of America.
  • D'Amours M; Hydra Biosciences, Cambridge, Massachusetts, United States of America.
  • Eickmeier C; Boehringer Ingelheim Pharma GmbH & Co. KG, Biberach an der Riss, Germany.
  • Fanger CM; Hydra Biosciences, Cambridge, Massachusetts, United States of America.
  • Hecker C; Boehringer Ingelheim Pharma GmbH & Co. KG, Biberach an der Riss, Germany.
  • Hessler DP; Hydra Biosciences, Cambridge, Massachusetts, United States of America.
  • Hengerer B; Boehringer Ingelheim Pharma GmbH & Co. KG, Biberach an der Riss, Germany.
  • Kroker KS; Boehringer Ingelheim Pharma GmbH & Co. KG, Biberach an der Riss, Germany.
  • Malekiani S; Hydra Biosciences, Cambridge, Massachusetts, United States of America.
  • Mihalek R; Hydra Biosciences, Cambridge, Massachusetts, United States of America.
  • McLaughlin J; Hydra Biosciences, Cambridge, Massachusetts, United States of America.
  • Rast G; Boehringer Ingelheim Pharma GmbH & Co. KG, Biberach an der Riss, Germany.
  • Witek J; Hydra Biosciences, Cambridge, Massachusetts, United States of America.
  • Sauer A; Boehringer Ingelheim Pharma GmbH & Co. KG, Biberach an der Riss, Germany.
  • Pryce CR; Preclinical Laboratory for Translational Research into Affective Disorders, Department of Psychiatry, Psychotherapy & Psychosomatics, Psychiatric Hospital, University of Zurich, Zurich, Switzerland.
  • Moran MM; Hydra Biosciences, Cambridge, Massachusetts, United States of America.
PLoS One ; 13(1): e0191225, 2018.
Article em En | MEDLINE | ID: mdl-29385160

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Ansiolíticos / Canais de Cátion TRPC / Compostos Heterocíclicos de 4 ou mais Anéis / Antidepressivos Limite: Animals / Humans Idioma: En Ano de publicação: 2018 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Ansiolíticos / Canais de Cátion TRPC / Compostos Heterocíclicos de 4 ou mais Anéis / Antidepressivos Limite: Animals / Humans Idioma: En Ano de publicação: 2018 Tipo de documento: Article