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Selective inhibition of human cathepsin S by 2,4,6-trisubstituted 1,3,5-triazine analogs.
Tber, Zahira; Wartenberg, Mylène; Jacques, Jean-Eddy; Roy, Vincent; Lecaille, Fabien; Warszycki, Dawid; Bojarski, Andrzej J; Lalmanach, Gilles; Agrofoglio, Luigi A.
Afiliação
  • Tber Z; Université d'Orléans, CNRS, ICOA, UMR 7311, F-45067 Orléans, France.
  • Wartenberg M; INSERM, UMR 1100, Centre d'Etude des Pathologies Respiratoires, Université François Rabelais, F-37032 Tours cedex, France.
  • Jacques JE; Université d'Orléans, CNRS, ICOA, UMR 7311, F-45067 Orléans, France.
  • Roy V; Université d'Orléans, CNRS, ICOA, UMR 7311, F-45067 Orléans, France. Electronic address: vincent.roy@univ-orleans.fr.
  • Lecaille F; INSERM, UMR 1100, Centre d'Etude des Pathologies Respiratoires, Université François Rabelais, F-37032 Tours cedex, France.
  • Warszycki D; Medicinal Chemistry Department, Institute of Pharmacology, Polish Academy of Sciences, Kraków, Poland.
  • Bojarski AJ; Medicinal Chemistry Department, Institute of Pharmacology, Polish Academy of Sciences, Kraków, Poland.
  • Lalmanach G; INSERM, UMR 1100, Centre d'Etude des Pathologies Respiratoires, Université François Rabelais, F-37032 Tours cedex, France.
  • Agrofoglio LA; Université d'Orléans, CNRS, ICOA, UMR 7311, F-45067 Orléans, France.
Bioorg Med Chem ; 26(14): 4310-4319, 2018 08 07.
Article em En | MEDLINE | ID: mdl-30049585

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Triazinas / Catepsinas / Inibidores Enzimáticos Limite: Humans Idioma: En Ano de publicação: 2018 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Triazinas / Catepsinas / Inibidores Enzimáticos Limite: Humans Idioma: En Ano de publicação: 2018 Tipo de documento: Article