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BRET-based assay to monitor EGFR transactivation by the AT1R reveals Gq/11 protein-independent activation and AT1R-EGFR complexes.
O'Brien, Shannon L; Johnstone, Elizabeth K M; Devost, Dominic; Conroy, Jacinta; Reichelt, Melissa E; Purdue, Brooke W; Ayoub, Mohammed A; Kawai, Tatsuo; Inoue, Asuka; Eguchi, Satoru; Hébert, Terence E; Pfleger, Kevin D G; Thomas, Walter G.
Afiliação
  • O'Brien SL; Receptor Biology Group, The School of Biomedical Sciences, Faculty of Medicine, The University of Queensland, St Lucia 4072, Queensland, Australia.
  • Johnstone EKM; Molecular Endocrinology and Pharmacology, Harry Perkins Institute of Medical Research, QEII Medical Centre, Nedlands and Centre for Medical Research, The University of Western Australia, Crawley, Western Australia 6009, Australia.
  • Devost D; Department of Pharmacology and Therapeutics, McGill University, Montreal, QC, Canada.
  • Conroy J; Receptor Biology Group, The School of Biomedical Sciences, Faculty of Medicine, The University of Queensland, St Lucia 4072, Queensland, Australia.
  • Reichelt ME; Receptor Biology Group, The School of Biomedical Sciences, Faculty of Medicine, The University of Queensland, St Lucia 4072, Queensland, Australia.
  • Purdue BW; Receptor Biology Group, The School of Biomedical Sciences, Faculty of Medicine, The University of Queensland, St Lucia 4072, Queensland, Australia.
  • Ayoub MA; Molecular Endocrinology and Pharmacology, Harry Perkins Institute of Medical Research, QEII Medical Centre, Nedlands and Centre for Medical Research, The University of Western Australia, Crawley, Western Australia 6009, Australia.
  • Kawai T; Cardiovascular Research Centre, Department of Physiology, Lewis Katz School of Medicine at Temple University, Philadelphia, PA, United States.
  • Inoue A; Graduate School of Pharmaceutical Sciences, Tohoku University, Sendai, Miyagi 980-8578, Japan.
  • Eguchi S; Cardiovascular Research Centre, Department of Physiology, Lewis Katz School of Medicine at Temple University, Philadelphia, PA, United States.
  • Hébert TE; Department of Pharmacology and Therapeutics, McGill University, Montreal, QC, Canada.
  • Pfleger KDG; Molecular Endocrinology and Pharmacology, Harry Perkins Institute of Medical Research, QEII Medical Centre, Nedlands and Centre for Medical Research, The University of Western Australia, Crawley, Western Australia 6009, Australia; Dimerix Limited, Nedlands, Western Australia 6009, Australia.
  • Thomas WG; Receptor Biology Group, The School of Biomedical Sciences, Faculty of Medicine, The University of Queensland, St Lucia 4072, Queensland, Australia; Centre for Cardiac and Vasculature Biology, The University of Queensland, St Lucia 4072, Queensland, Australia. Electronic address: w.thomas@uq.edu.au.
Biochem Pharmacol ; 158: 232-242, 2018 12.
Article em En | MEDLINE | ID: mdl-30347205

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Ativação Transcricional / Subunidades alfa Gq-G11 de Proteínas de Ligação ao GTP / Receptor Tipo 1 de Angiotensina / Técnicas de Transferência de Energia por Ressonância de Bioluminescência Limite: Animals / Humans / Male Idioma: En Ano de publicação: 2018 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Ativação Transcricional / Subunidades alfa Gq-G11 de Proteínas de Ligação ao GTP / Receptor Tipo 1 de Angiotensina / Técnicas de Transferência de Energia por Ressonância de Bioluminescência Limite: Animals / Humans / Male Idioma: En Ano de publicação: 2018 Tipo de documento: Article