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Selective inhibition of carbonic anhydrase IX over carbonic anhydrase XII in breast cancer cells using benzene sulfonamides: Disconnect between activity and growth inhibition.
Mboge, Mam Y; Chen, Zhijuan; Wolff, Alyssa; Mathias, John V; Tu, Chingkuang; Brown, Kevin D; Bozdag, Murat; Carta, Fabrizio; Supuran, Claudiu T; McKenna, Robert; Frost, Susan C.
Afiliação
  • Mboge MY; Department of Biochemistry and Molecular Biology, University of Florida, Gainesville, FL, United States of America.
  • Chen Z; Department of Biochemistry and Molecular Biology, University of Florida, Gainesville, FL, United States of America.
  • Wolff A; Department of Biochemistry and Molecular Biology, University of Florida, Gainesville, FL, United States of America.
  • Mathias JV; Department of Biochemistry and Molecular Biology, University of Florida, Gainesville, FL, United States of America.
  • Tu C; Department of Biochemistry and Molecular Biology, University of Florida, Gainesville, FL, United States of America.
  • Brown KD; Department of Biochemistry and Molecular Biology, University of Florida, Gainesville, FL, United States of America.
  • Bozdag M; University of Florence, NEUROFARBA Department, Sezione di Farmaceutica e Nutraceutica, Sesto Fiorentino (Florence), Italy.
  • Carta F; University of Florence, NEUROFARBA Department, Sezione di Farmaceutica e Nutraceutica, Sesto Fiorentino (Florence), Italy.
  • Supuran CT; University of Florence, NEUROFARBA Department, Sezione di Farmaceutica e Nutraceutica, Sesto Fiorentino (Florence), Italy.
  • McKenna R; Department of Biochemistry and Molecular Biology, University of Florida, Gainesville, FL, United States of America.
  • Frost SC; Department of Biochemistry and Molecular Biology, University of Florida, Gainesville, FL, United States of America.
PLoS One ; 13(11): e0207417, 2018.
Article em En | MEDLINE | ID: mdl-30452451

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Sulfonamidas / Derivados de Benzeno / Neoplasias da Mama / Inibidores da Anidrase Carbônica / Anidrases Carbônicas / Anidrase Carbônica IX / Antígenos de Neoplasias / Proteínas de Neoplasias Limite: Female / Humans Idioma: En Ano de publicação: 2018 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Sulfonamidas / Derivados de Benzeno / Neoplasias da Mama / Inibidores da Anidrase Carbônica / Anidrases Carbônicas / Anidrase Carbônica IX / Antígenos de Neoplasias / Proteínas de Neoplasias Limite: Female / Humans Idioma: En Ano de publicação: 2018 Tipo de documento: Article