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Synthesis and anti-tumor activity of imidazopyrazines as TAK1 inhibitors.
Kang, Seok Jong; Lee, Jung Wuk; Chung, Shin Hyuck; Jang, Sun Young; Choi, Jaeyul; Suh, Kwee Hyun; Kim, Young Hoon; Ham, Young Jin; Min, Kyung Hoon.
Afiliação
  • Kang SJ; College of Pharmacy, Chung-Ang University, Seoul, 06974, Republic of Korea; Department of Drug Discovery, Hanmi Research Center, Gyeonggi-do, 18469, Republic of Korea.
  • Lee JW; College of Pharmacy, Chung-Ang University, Seoul, 06974, Republic of Korea.
  • Chung SH; College of Pharmacy, Chung-Ang University, Seoul, 06974, Republic of Korea.
  • Jang SY; College of Pharmacy, Chung-Ang University, Seoul, 06974, Republic of Korea; Department of Drug Discovery, Hanmi Research Center, Gyeonggi-do, 18469, Republic of Korea.
  • Choi J; Department of Drug Discovery, Hanmi Research Center, Gyeonggi-do, 18469, Republic of Korea.
  • Suh KH; Department of Drug Discovery, Hanmi Research Center, Gyeonggi-do, 18469, Republic of Korea.
  • Kim YH; Department of Drug Discovery, Hanmi Research Center, Gyeonggi-do, 18469, Republic of Korea.
  • Ham YJ; Department of Drug Discovery, Hanmi Research Center, Gyeonggi-do, 18469, Republic of Korea.
  • Min KH; College of Pharmacy, Chung-Ang University, Seoul, 06974, Republic of Korea. Electronic address: khmin@cau.ac.kr.
Eur J Med Chem ; 163: 660-670, 2019 Feb 01.
Article em En | MEDLINE | ID: mdl-30576901

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Pirazinas / MAP Quinase Quinase Quinases / Inibidores de Proteínas Quinases Limite: Animals / Humans Idioma: En Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Pirazinas / MAP Quinase Quinase Quinases / Inibidores de Proteínas Quinases Limite: Animals / Humans Idioma: En Ano de publicação: 2019 Tipo de documento: Article