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Design, synthesis and biological evaluation of certain CDK2 inhibitors based on pyrazole and pyrazolo[1,5-a] pyrimidine scaffold with apoptotic activity.
Ali, Ghada M E; Ibrahim, Diaa A; Elmetwali, Amira M; Ismail, Nasser S M.
Afiliação
  • Ali GME; National Organization for Drug Control & Research, P.O. Box: 29, Cairo, Egypt.
  • Ibrahim DA; National Organization for Drug Control & Research, P.O. Box: 29, Cairo, Egypt.
  • Elmetwali AM; National Organization for Drug Control & Research, P.O. Box: 29, Cairo, Egypt.
  • Ismail NSM; Pharmaceutical Chemistry Department, Faculty of Pharmaceutical Sciences and Pharmaceutical Industries, Future University in Egypt, Cairo 12311, Egypt. Electronic address: saadnasser2003@yahoo.com.
Bioorg Chem ; 86: 1-14, 2019 05.
Article em En | MEDLINE | ID: mdl-30682722

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Pirazóis / Pirimidinas / Desenho de Fármacos / Apoptose / Inibidores de Proteínas Quinases / Quinase 2 Dependente de Ciclina / Antineoplásicos Limite: Humans Idioma: En Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Pirazóis / Pirimidinas / Desenho de Fármacos / Apoptose / Inibidores de Proteínas Quinases / Quinase 2 Dependente de Ciclina / Antineoplásicos Limite: Humans Idioma: En Ano de publicação: 2019 Tipo de documento: Article