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Pharmacophore-guided discovery of CDC25 inhibitors causing cell cycle arrest and tumor regression.
Kabakci, Zeynep; Käppeli, Simon; Cantù, Claudio; Jensen, Lasse D; König, Christiane; Toggweiler, Janine; Gentili, Christian; Ribaudo, Giovanni; Zagotto, Giuseppe; Basler, Konrad; Pinna, Lorenzo A; Cozza, Giorgio; Ferrari, Stefano.
Afiliação
  • Kabakci Z; Institute of Molecular Cancer Research, University of Zurich, Winterthurerstrasse 190, CH-8057, Zurich, Switzerland.
  • Käppeli S; Institute of Molecular Cancer Research, University of Zurich, Winterthurerstrasse 190, CH-8057, Zurich, Switzerland.
  • Cantù C; Department of Clinical and Experimental Medicine, Campus US, University of Linköping, S-58183, Linköping, Sweden.
  • Jensen LD; Wallenberg Centre for Molecular Medicine, University of Linköping, S-58183, Linköping, Sweden.
  • König C; Institute of Molecular Life Sciences, University of Zurich, Winterthurerstrasse 190, CH-8057, Zurich, Switzerland.
  • Toggweiler J; Department of Medical and Health Sciences, Campus US, University of Linköping, S-58183, Linköping, Sweden.
  • Gentili C; Institute of Molecular Cancer Research, University of Zurich, Winterthurerstrasse 190, CH-8057, Zurich, Switzerland.
  • Ribaudo G; Institute of Molecular Life Sciences, University of Zurich, Winterthurerstrasse 190, CH-8057, Zurich, Switzerland.
  • Zagotto G; Institute of Molecular Cancer Research, University of Zurich, Winterthurerstrasse 190, CH-8057, Zurich, Switzerland.
  • Basler K; Department of Pharmacology, University of Padua, Via U. Bassi 58/B, I-35131, Padua, Italy.
  • Pinna LA; Department of Pharmacology, University of Padua, Via U. Bassi 58/B, I-35131, Padua, Italy.
  • Cozza G; Institute of Molecular Life Sciences, University of Zurich, Winterthurerstrasse 190, CH-8057, Zurich, Switzerland.
  • Ferrari S; Department of Biomedical Sciences, University of Padua, Via U. Bassi 58/B, I-35131, Padua, Italy.
Sci Rep ; 9(1): 1335, 2019 02 04.
Article em En | MEDLINE | ID: mdl-30718768

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Conformação Proteica / Proteína Quinase CDC2 / Fosfatases cdc25 / Neoplasias Limite: Animals / Humans Idioma: En Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Conformação Proteica / Proteína Quinase CDC2 / Fosfatases cdc25 / Neoplasias Limite: Animals / Humans Idioma: En Ano de publicação: 2019 Tipo de documento: Article