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A comparative study of the binding properties, dipeptidyl peptidase-4 (DPP-4) inhibitory activity and glucose-lowering efficacy of the DPP-4 inhibitors alogliptin, linagliptin, saxagliptin, sitagliptin and vildagliptin in mice.
Berger, Joel P; SinhaRoy, Ranabir; Pocai, Alessandro; Kelly, Theresa M; Scapin, Giovanna; Gao, Ying-Duo; Pryor, Kelly Ann D; Wu, Joseph K; Eiermann, George J; Xu, Shiyao S; Zhang, Xiaoping; Tatosian, Daniel A; Weber, Ann E; Thornberry, Nancy A; Carr, Richard D.
Afiliação
  • Berger JP; Merck& Co., Inc. Kenilworth NJ USA.
  • SinhaRoy R; Present address: Takeda Pharmaceuticals International, Inc. Cambridge MA USA.
  • Pocai A; Merck& Co., Inc. Kenilworth NJ USA.
  • Kelly TM; Present address: Janssen Pharmaceuticals, Inc. Titusville NJ USA.
  • Scapin G; Merck& Co., Inc. Kenilworth NJ USA.
  • Gao YD; Present address: Janssen Pharmaceuticals, Inc. Titusville NJ USA.
  • Pryor KAD; Merck& Co., Inc. Kenilworth NJ USA.
  • Wu JK; Merck& Co., Inc. Kenilworth NJ USA.
  • Eiermann GJ; Merck& Co., Inc. Kenilworth NJ USA.
  • Xu SS; Merck& Co., Inc. Kenilworth NJ USA.
  • Zhang X; Merck& Co., Inc. Kenilworth NJ USA.
  • Tatosian DA; Merck& Co., Inc. Kenilworth NJ USA.
  • Weber AE; Merck& Co., Inc. Kenilworth NJ USA.
  • Thornberry NA; Merck& Co., Inc. Kenilworth NJ USA.
  • Carr RD; Merck& Co., Inc. Kenilworth NJ USA.
Endocrinol Diabetes Metab ; 1(1): e00002, 2018 Jan.
Article em En | MEDLINE | ID: mdl-30815539

Texto completo: 1 Base de dados: MEDLINE Idioma: En Ano de publicação: 2018 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Idioma: En Ano de publicação: 2018 Tipo de documento: Article