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Clathrin and GRK2/3 inhibitors block δ-opioid receptor internalization in myenteric neurons and inhibit neuromuscular transmission in the mouse colon.
DiCello, Jesse J; Rajasekhar, Pradeep; Eriksson, Emily M; Saito, Ayame; Gondin, Arisbel B; Veldhuis, Nicholas A; Canals, Meritxell; Carbone, Simona E; Poole, Daniel P.
Afiliação
  • DiCello JJ; Drug Discovery Biology Theme, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.
  • Rajasekhar P; ARC Centre of Excellence in Convergent Bio-Nano Science and Technology, Parkville, Victoria, Australia.
  • Eriksson EM; Drug Discovery Biology Theme, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.
  • Saito A; Divisions of Population Health & Immunity and Infection and Immunity, The Walter and Eliza Hall Institute, Parkville, Victoria, Australia.
  • Gondin AB; Department of Medical Biology, The University of Melbourne, Parkville, Victoria, Australia.
  • Veldhuis NA; Drug Discovery Biology Theme, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.
  • Canals M; ARC Centre of Excellence in Convergent Bio-Nano Science and Technology, Parkville, Victoria, Australia.
  • Carbone SE; Drug Discovery Biology Theme, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.
  • Poole DP; ARC Centre of Excellence in Convergent Bio-Nano Science and Technology, Parkville, Victoria, Australia.
Am J Physiol Gastrointest Liver Physiol ; 317(2): G79-G89, 2019 08 01.
Article em En | MEDLINE | ID: mdl-31091149

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Piridinas / Sulfonamidas / Triazóis / Benzamidas / Clatrina / Colo / Receptores Opioides delta / Endocitose / Tiazolidinas / Músculo Liso Limite: Animals Idioma: En Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Piridinas / Sulfonamidas / Triazóis / Benzamidas / Clatrina / Colo / Receptores Opioides delta / Endocitose / Tiazolidinas / Músculo Liso Limite: Animals Idioma: En Ano de publicação: 2019 Tipo de documento: Article