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BRD4 bimodal binding at promoters and drug-induced displacement at Pol II pause sites associates with I-BET sensitivity.
Khoueiry, P; Ward Gahlawat, A; Petretich, M; Michon, A M; Simola, D; Lam, E; Furlong, E E; Benes, V; Dawson, M A; Prinjha, R K; Drewes, G; Grandi, P.
Afiliação
  • Khoueiry P; Cellzome GmbH, a GSK Company, Heidelberg, Germany. pk17@aub.edu.lb.
  • Ward Gahlawat A; Department of Biochemistry and Molecular Genetics, Faculty of Medicine, American University of Beirut, Beirut, Lebanon. pk17@aub.edu.lb.
  • Petretich M; Cellzome GmbH, a GSK Company, Heidelberg, Germany.
  • Michon AM; Cellzome GmbH, a GSK Company, Heidelberg, Germany.
  • Simola D; Cellzome GmbH, a GSK Company, Heidelberg, Germany.
  • Lam E; Target Science Computational Biology, GSK Medicines Research Centre, Upper Providence, USA.
  • Furlong EE; Peter MacCallum Cancer Center, Melbourne, Australia.
  • Benes V; European Molecular Biology Laboratory (EMBL), Genome Biology Unit, Heidelberg, Germany.
  • Dawson MA; European Molecular Biology Laboratory (EMBL), Genomics Core Facility, Heidelberg, Germany.
  • Prinjha RK; Peter MacCallum Cancer Center, Melbourne, Australia.
  • Drewes G; Epigenetics DPU, GSK Medicines Research Centre, Stevenage, UK.
  • Grandi P; Cellzome GmbH, a GSK Company, Heidelberg, Germany.
Epigenetics Chromatin ; 12(1): 39, 2019 07 02.
Article em En | MEDLINE | ID: mdl-31266503

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Fatores de Transcrição / RNA Polimerase II / Proteínas / Proteínas de Ciclo Celular / Compostos Heterocíclicos de 4 ou mais Anéis Tipo de estudo: Diagnostic_studies / Prognostic_studies / Risk_factors_studies Limite: Humans Idioma: En Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Fatores de Transcrição / RNA Polimerase II / Proteínas / Proteínas de Ciclo Celular / Compostos Heterocíclicos de 4 ou mais Anéis Tipo de estudo: Diagnostic_studies / Prognostic_studies / Risk_factors_studies Limite: Humans Idioma: En Ano de publicação: 2019 Tipo de documento: Article