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Development and Validation of a Higher-Throughput Cytochrome P450 Inhibition Assay with the Novel Cofactor-Supplemented Permeabilized Cryopreserved Human Hepatocytes (MetMax Human Hepatocytes).
Palacharla, Veera Raghava Choudary; Chunduru, Prathyusha; Ajjala, Devender Reddy; Bhyrapuneni, Gopinadh; Nirogi, Ramakrishna; Li, Albert P.
Afiliação
  • Palacharla VRC; Drug Metabolism and Pharmacokinetics, Suven Life Sciences Ltd., Jeedimetla, Hyderabad, India (V.R.C.P., G.B., R.N.); Bio-analysis, Suven Life Sciences Ltd., Pashamylaram, Medak, India (P.C., D.R.A.); and In Vitro ADMET Laboratories Inc., Columbia, Maryland (A.P.L.).
  • Chunduru P; Drug Metabolism and Pharmacokinetics, Suven Life Sciences Ltd., Jeedimetla, Hyderabad, India (V.R.C.P., G.B., R.N.); Bio-analysis, Suven Life Sciences Ltd., Pashamylaram, Medak, India (P.C., D.R.A.); and In Vitro ADMET Laboratories Inc., Columbia, Maryland (A.P.L.).
  • Ajjala DR; Drug Metabolism and Pharmacokinetics, Suven Life Sciences Ltd., Jeedimetla, Hyderabad, India (V.R.C.P., G.B., R.N.); Bio-analysis, Suven Life Sciences Ltd., Pashamylaram, Medak, India (P.C., D.R.A.); and In Vitro ADMET Laboratories Inc., Columbia, Maryland (A.P.L.).
  • Bhyrapuneni G; Drug Metabolism and Pharmacokinetics, Suven Life Sciences Ltd., Jeedimetla, Hyderabad, India (V.R.C.P., G.B., R.N.); Bio-analysis, Suven Life Sciences Ltd., Pashamylaram, Medak, India (P.C., D.R.A.); and In Vitro ADMET Laboratories Inc., Columbia, Maryland (A.P.L.).
  • Nirogi R; Drug Metabolism and Pharmacokinetics, Suven Life Sciences Ltd., Jeedimetla, Hyderabad, India (V.R.C.P., G.B., R.N.); Bio-analysis, Suven Life Sciences Ltd., Pashamylaram, Medak, India (P.C., D.R.A.); and In Vitro ADMET Laboratories Inc., Columbia, Maryland (A.P.L.) nvsrk@suven.com.
  • Li AP; Drug Metabolism and Pharmacokinetics, Suven Life Sciences Ltd., Jeedimetla, Hyderabad, India (V.R.C.P., G.B., R.N.); Bio-analysis, Suven Life Sciences Ltd., Pashamylaram, Medak, India (P.C., D.R.A.); and In Vitro ADMET Laboratories Inc., Columbia, Maryland (A.P.L.) lialbert@invitroadmet.com.
Drug Metab Dispos ; 47(10): 1032-1039, 2019 10.
Article em En | MEDLINE | ID: mdl-31375472

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Técnicas de Cultura de Células / Sistema Enzimático do Citocromo P-450 / Ensaios Enzimáticos / Ensaios de Triagem em Larga Escala / Inibidores das Enzimas do Citocromo P-450 Limite: Humans Idioma: En Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Técnicas de Cultura de Células / Sistema Enzimático do Citocromo P-450 / Ensaios Enzimáticos / Ensaios de Triagem em Larga Escala / Inibidores das Enzimas do Citocromo P-450 Limite: Humans Idioma: En Ano de publicação: 2019 Tipo de documento: Article