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Data-Driven Construction of Antitumor Agents with Controlled Polypharmacology.
Da, Chenxiao; Zhang, Dehui; Stashko, Michael; Vasileiadi, Eleana; Parker, Rebecca E; Minson, Katherine A; Huey, Madeline G; Huelse, Justus M; Hunter, Debra; Gilbert, Thomas S K; Norris-Drouin, Jacqueline; Miley, Michael; Herring, Laura E; Graves, Lee M; DeRyckere, Deborah; Earp, H Shelton; Graham, Douglas K; Frye, Stephen V; Wang, Xiaodong; Kireev, Dmitri.
Afiliação
  • Da C; Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology and Medicinal Chemistry, Eshelman School of Pharmacy , University of North Carolina at Chapel Hill , Chapel Hill , North Carolina 27599-7363 , United States.
  • Zhang D; Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology and Medicinal Chemistry, Eshelman School of Pharmacy , University of North Carolina at Chapel Hill , Chapel Hill , North Carolina 27599-7363 , United States.
  • Stashko M; Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology and Medicinal Chemistry, Eshelman School of Pharmacy , University of North Carolina at Chapel Hill , Chapel Hill , North Carolina 27599-7363 , United States.
  • Vasileiadi E; Aflac Cancer and Blood Disorders Center, Children's Healthcare of Atlanta, and Department of Pediatrics , Emory University , Atlanta , Georgia 30322 , United States.
  • Parker RE; Aflac Cancer and Blood Disorders Center, Children's Healthcare of Atlanta, and Department of Pediatrics , Emory University , Atlanta , Georgia 30322 , United States.
  • Minson KA; Aflac Cancer and Blood Disorders Center, Children's Healthcare of Atlanta, and Department of Pediatrics , Emory University , Atlanta , Georgia 30322 , United States.
  • Huey MG; Aflac Cancer and Blood Disorders Center, Children's Healthcare of Atlanta, and Department of Pediatrics , Emory University , Atlanta , Georgia 30322 , United States.
  • Huelse JM; Aflac Cancer and Blood Disorders Center, Children's Healthcare of Atlanta, and Department of Pediatrics , Emory University , Atlanta , Georgia 30322 , United States.
  • Norris-Drouin J; Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology and Medicinal Chemistry, Eshelman School of Pharmacy , University of North Carolina at Chapel Hill , Chapel Hill , North Carolina 27599-7363 , United States.
  • DeRyckere D; Aflac Cancer and Blood Disorders Center, Children's Healthcare of Atlanta, and Department of Pediatrics , Emory University , Atlanta , Georgia 30322 , United States.
  • Graham DK; Aflac Cancer and Blood Disorders Center, Children's Healthcare of Atlanta, and Department of Pediatrics , Emory University , Atlanta , Georgia 30322 , United States.
  • Frye SV; Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology and Medicinal Chemistry, Eshelman School of Pharmacy , University of North Carolina at Chapel Hill , Chapel Hill , North Carolina 27599-7363 , United States.
  • Wang X; Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology and Medicinal Chemistry, Eshelman School of Pharmacy , University of North Carolina at Chapel Hill , Chapel Hill , North Carolina 27599-7363 , United States.
  • Kireev D; Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology and Medicinal Chemistry, Eshelman School of Pharmacy , University of North Carolina at Chapel Hill , Chapel Hill , North Carolina 27599-7363 , United States.
J Am Chem Soc ; 141(39): 15700-15709, 2019 10 02.
Article em En | MEDLINE | ID: mdl-31497954

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Receptores Proteína Tirosina Quinases / Antineoplásicos Limite: Animals / Humans Idioma: En Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Receptores Proteína Tirosina Quinases / Antineoplásicos Limite: Animals / Humans Idioma: En Ano de publicação: 2019 Tipo de documento: Article