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Preclinical In Vitro and In Vivo Characterization of Synaptic Vesicle 2A-Targeting Compounds Amenable to F-18 Labeling as Potential PET Radioligands for Imaging of Synapse Integrity.
Patel, Shil; Knight, Ashley; Krause, Stephen; Teceno, Tyler; Tresse, Cedric; Li, Songye; Cai, Zhengxin; Gouasmat, Alexandra; Carroll, Vincent M; Barret, Olivier; Gottmukkala, Vijay; Zhang, Wenjie; Xiang, Xianhong; Morley, Thomas; Huang, Yiyun; Passchier, Jan.
Afiliação
  • Patel S; Codiak Biosciences, 500 Technology Square, 9th Floor, Cambridge, MA, 02139, USA. shil.patel@codiakbio.com.
  • Knight A; Centre for Addiction and Mental Health, University of Toronto, 250 College Street, Toronto, ON, M5T 1R8, Canada.
  • Krause S; Eisai Inc., 100 Tice Blvd, Woodcliff Lake, NJ, 07677, USA.
  • Teceno T; Eisai Inc., 100 Tice Blvd, Woodcliff Lake, NJ, 07677, USA.
  • Tresse C; Invicro, LLC, 27 Drydock Ave. 7th Floor West, Boston, MA, 02210, USA.
  • Li S; PET Center, Department of Radiology and Biomedical Imaging, Yale University School of Medicine, 801 Howard Avenue, New Haven, CT, 06510, USA.
  • Cai Z; PET Center, Department of Radiology and Biomedical Imaging, Yale University School of Medicine, 801 Howard Avenue, New Haven, CT, 06510, USA.
  • Gouasmat A; Invicro, LLC, 27 Drydock Ave. 7th Floor West, Boston, MA, 02210, USA.
  • Carroll VM; Invicro, LLC, 27 Drydock Ave. 7th Floor West, Boston, MA, 02210, USA.
  • Barret O; Invicro, LLC, 27 Drydock Ave. 7th Floor West, Boston, MA, 02210, USA.
  • Gottmukkala V; Invicro, LLC, 27 Drydock Ave. 7th Floor West, Boston, MA, 02210, USA.
  • Zhang W; Department of Nuclear Medicine, West China Hospital, Sichuan University, Chengdu, 610041, Sichuan, China.
  • Xiang X; Department of Interventional Radiology, The First Affiliated Hospital of Sun Yat-Sen University, 58 Zhongshan Second Road, Yuexiu District, Guangzhou, 510080, China.
  • Morley T; Invicro, LLC, 27 Drydock Ave. 7th Floor West, Boston, MA, 02210, USA.
  • Huang Y; PET Center, Department of Radiology and Biomedical Imaging, Yale University School of Medicine, 801 Howard Avenue, New Haven, CT, 06510, USA.
  • Passchier J; Invicro, LLC, 27 Drydock Ave. 7th Floor West, Boston, MA, 02210, USA.
Mol Imaging Biol ; 22(4): 832-841, 2020 08.
Article em En | MEDLINE | ID: mdl-31728839

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Coloração e Rotulagem / Sinapses / Radioisótopos de Flúor / Glicoproteínas de Membrana / Compostos Radiofarmacêuticos / Proteínas do Tecido Nervoso Tipo de estudo: Prognostic_studies Limite: Animals / Humans Idioma: En Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Coloração e Rotulagem / Sinapses / Radioisótopos de Flúor / Glicoproteínas de Membrana / Compostos Radiofarmacêuticos / Proteínas do Tecido Nervoso Tipo de estudo: Prognostic_studies Limite: Animals / Humans Idioma: En Ano de publicação: 2020 Tipo de documento: Article