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Investigation of the Adrenergic and Opioid Binding Affinities, Metabolic Stability, Plasma Protein Binding Properties, and Functional Effects of Selected Indole-Based Kratom Alkaloids.
Obeng, Samuel; Kamble, Shyam H; Reeves, Morgan E; Restrepo, Luis F; Patel, Avi; Behnke, Mira; Chear, Nelson J-Y; Ramanathan, Surash; Sharma, Abhisheak; León, Francisco; Hiranita, Takato; Avery, Bonnie A; McMahon, Lance R; McCurdy, Christopher R.
Afiliação
  • Obeng S; Department of Pharmacodynamics, College of Pharmacy , University of Florida , Gainesville , Florida 32610 , United States.
  • Kamble SH; Department of Medicinal Chemistry , College of Pharmacy, University of Florida , Gainesville , Florida 32610 , United States.
  • Reeves ME; Department of Pharmaceutics, College of Pharmacy , University of Florida , Gainesville , Florida 32610 , United States.
  • Restrepo LF; Translational Drug Development Core, Clinical and Translational Sciences Institute , University of Florida , Gainesville , Florida 32610 , United States.
  • Patel A; Department of Pharmacodynamics, College of Pharmacy , University of Florida , Gainesville , Florida 32610 , United States.
  • Behnke M; Department of Pharmacodynamics, College of Pharmacy , University of Florida , Gainesville , Florida 32610 , United States.
  • Chear NJ; Department of Pharmacodynamics, College of Pharmacy , University of Florida , Gainesville , Florida 32610 , United States.
  • Ramanathan S; Department of Pharmacodynamics, College of Pharmacy , University of Florida , Gainesville , Florida 32610 , United States.
  • Sharma A; Centre for Drug Research , Universiti Sains Malaysia , 11800 Minden , Penang , Malaysia.
  • León F; Centre for Drug Research , Universiti Sains Malaysia , 11800 Minden , Penang , Malaysia.
  • Hiranita T; Department of Pharmaceutics, College of Pharmacy , University of Florida , Gainesville , Florida 32610 , United States.
  • Avery BA; Translational Drug Development Core, Clinical and Translational Sciences Institute , University of Florida , Gainesville , Florida 32610 , United States.
  • McMahon LR; Department of Medicinal Chemistry , College of Pharmacy, University of Florida , Gainesville , Florida 32610 , United States.
  • McCurdy CR; Department of Pharmacodynamics, College of Pharmacy , University of Florida , Gainesville , Florida 32610 , United States.
J Med Chem ; 63(1): 433-439, 2020 01 09.
Article em En | MEDLINE | ID: mdl-31834797

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Proteínas Sanguíneas / Dopaminérgicos / Adrenérgicos / Alcaloides de Triptamina e Secologanina / Analgésicos Limite: Animals / Humans Idioma: En Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Proteínas Sanguíneas / Dopaminérgicos / Adrenérgicos / Alcaloides de Triptamina e Secologanina / Analgésicos Limite: Animals / Humans Idioma: En Ano de publicação: 2020 Tipo de documento: Article