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Negative allosteric modulators of the human calcium-sensing receptor bind to overlapping and distinct sites within the 7-transmembrane domain.
Josephs, Tracy M; Keller, Andrew N; Khajehali, Elham; DeBono, Aaron; Langmead, Christopher J; Conigrave, Arthur D; Capuano, Ben; Kufareva, Irina; Gregory, Karen J; Leach, Katie.
Afiliação
  • Josephs TM; Drug Discovery Biology and Department of Pharmacology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.
  • Keller AN; Drug Discovery Biology and Department of Pharmacology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.
  • Khajehali E; Drug Discovery Biology and Department of Pharmacology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.
  • DeBono A; Drug Discovery Biology and Department of Pharmacology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.
  • Langmead CJ; Drug Discovery Biology and Department of Pharmacology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.
  • Conigrave AD; School of Life and Environmental Sciences, University of Sydney, Sydney, NSW, Australia.
  • Capuano B; Drug Discovery Biology and Department of Pharmacology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.
  • Kufareva I; Skaggs School of Pharmacy & Pharmaceutical Sciences, University of California, San Diego, CA, USA.
  • Gregory KJ; Drug Discovery Biology and Department of Pharmacology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.
  • Leach K; Drug Discovery Biology and Department of Pharmacology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.
Br J Pharmacol ; 177(8): 1917-1930, 2020 04.
Article em En | MEDLINE | ID: mdl-31881094

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Receptores de Detecção de Cálcio Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Receptores de Detecção de Cálcio Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Ano de publicação: 2020 Tipo de documento: Article