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New 2-Ethylthio-4-methylaminoquinazoline derivatives inhibiting two subunits of cytochrome bc1 in Mycobacterium tuberculosis.
Lupien, Andréanne; Foo, Caroline Shi-Yan; Savina, Svetlana; Vocat, Anthony; Piton, Jérémie; Monakhova, Natalia; Benjak, Andrej; Lamprecht, Dirk A; Steyn, Adrie J C; Pethe, Kevin; Makarov, Vadim A; Cole, Stewart T.
Afiliação
  • Lupien A; Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland.
  • Foo CS; Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland.
  • Savina S; Department of Stresses of Microorganisms, A. N. Bach Institute of Biochemistry, Moscow, Russian Federation.
  • Vocat A; Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland.
  • Piton J; Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland.
  • Monakhova N; Department of Stresses of Microorganisms, A. N. Bach Institute of Biochemistry, Moscow, Russian Federation.
  • Benjak A; Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland.
  • Lamprecht DA; Africa Health Research Institute, Durban, South Africa.
  • Steyn AJC; Africa Health Research Institute, Durban, South Africa.
  • Pethe K; Department of Microbiology, University of Alabama at Birmingham, Birmingham, Alabama, United States of America.
  • Makarov VA; Lee Kong Chian School of Medicine and School of Biological Sciences, Nanyang Technological University, Singapore.
  • Cole ST; Department of Stresses of Microorganisms, A. N. Bach Institute of Biochemistry, Moscow, Russian Federation.
PLoS Pathog ; 16(1): e1008270, 2020 01.
Article em En | MEDLINE | ID: mdl-31971990

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Quinazolinas / Proteínas de Bactérias / Tuberculose Resistente a Múltiplos Medicamentos / Complexo III da Cadeia de Transporte de Elétrons / Mycobacterium tuberculosis / Antituberculosos Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Quinazolinas / Proteínas de Bactérias / Tuberculose Resistente a Múltiplos Medicamentos / Complexo III da Cadeia de Transporte de Elétrons / Mycobacterium tuberculosis / Antituberculosos Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Ano de publicação: 2020 Tipo de documento: Article