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A novel series of cysteine-dependent, allosteric inverse agonists of the nuclear receptor RORγt.
Jiang, Xin; Dulubova, Irina; Reisman, Scott A; Hotema, Martha; Lee, Chun-Yue I; Liu, Liping; McCauley, Lyndsey; Trevino, Isaac; Ferguson, Deborah A; Eken, Yigitcan; Wilson, Angela K; Wigley, W Christian; Visnick, Melean.
Afiliação
  • Jiang X; Reata Pharmaceuticals, Inc., 2801 Gateway Drive, Suite 150, Irving, TX 75063, USA.
  • Dulubova I; Reata Pharmaceuticals, Inc., 2801 Gateway Drive, Suite 150, Irving, TX 75063, USA.
  • Reisman SA; Reata Pharmaceuticals, Inc., 2801 Gateway Drive, Suite 150, Irving, TX 75063, USA.
  • Hotema M; Reata Pharmaceuticals, Inc., 2801 Gateway Drive, Suite 150, Irving, TX 75063, USA.
  • Lee CI; Reata Pharmaceuticals, Inc., 2801 Gateway Drive, Suite 150, Irving, TX 75063, USA.
  • Liu L; Reata Pharmaceuticals, Inc., 2801 Gateway Drive, Suite 150, Irving, TX 75063, USA.
  • McCauley L; Reata Pharmaceuticals, Inc., 2801 Gateway Drive, Suite 150, Irving, TX 75063, USA.
  • Trevino I; Reata Pharmaceuticals, Inc., 2801 Gateway Drive, Suite 150, Irving, TX 75063, USA.
  • Ferguson DA; Reata Pharmaceuticals, Inc., 2801 Gateway Drive, Suite 150, Irving, TX 75063, USA.
  • Eken Y; Department of Chemistry, Michigan State University, 578 South Shaw Lane, East Lansing, MI 48824, USA.
  • Wilson AK; Department of Chemistry, Michigan State University, 578 South Shaw Lane, East Lansing, MI 48824, USA.
  • Wigley WC; Reata Pharmaceuticals, Inc., 2801 Gateway Drive, Suite 150, Irving, TX 75063, USA.
  • Visnick M; Reata Pharmaceuticals, Inc., 2801 Gateway Drive, Suite 150, Irving, TX 75063, USA. Electronic address: mike.visnick@reatapharma.com.
Bioorg Med Chem Lett ; 30(6): 126967, 2020 03 15.
Article em En | MEDLINE | ID: mdl-32005415

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Artrite Reumatoide / Pirimidinas / Cisteína / Membro 3 do Grupo F da Subfamília 1 de Receptores Nucleares Limite: Animals / Humans Idioma: En Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Artrite Reumatoide / Pirimidinas / Cisteína / Membro 3 do Grupo F da Subfamília 1 de Receptores Nucleares Limite: Animals / Humans Idioma: En Ano de publicação: 2020 Tipo de documento: Article