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Characterization of Specific N-α-Acetyltransferase 50 (Naa50) Inhibitors Identified Using a DNA Encoded Library.
Kung, Pei-Pei; Bingham, Patrick; Burke, Benjamin J; Chen, Qiuxia; Cheng, Xuemin; Deng, Ya-Li; Dou, Dengfeng; Feng, Junli; Gallego, Gary M; Gehring, Michael R; Grant, Stephan K; Greasley, Samantha; Harris, Anthony R; Maegley, Karen A; Meier, Jordan; Meng, Xiaoyun; Montano, Jose L; Morgan, Barry A; Naughton, Brigitte S; Palde, Prakash B; Paul, Thomas A; Richardson, Paul; Sakata, Sylvie; Shaginian, Alex; Sonnenburg, William K; Subramanyam, Chakrapani; Timofeevski, Sergei; Wan, Jinqiao; Yan, Wen; Stewart, Albert E.
Afiliação
  • Kung PP; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.
  • Bingham P; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.
  • Burke BJ; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.
  • Chen Q; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China.
  • Cheng X; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China.
  • Deng YL; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.
  • Dou D; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China.
  • Feng J; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.
  • Gallego GM; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.
  • Gehring MR; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.
  • Grant SK; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.
  • Greasley S; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.
  • Harris AR; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.
  • Maegley KA; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.
  • Meier J; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States.
  • Meng X; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China.
  • Montano JL; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States.
  • Morgan BA; HitGen Pharmaceuticals Inc., PO Box 88240, Houston, Texas 77288, United States.
  • Naughton BS; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China.
  • Palde PB; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.
  • Paul TA; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.
  • Richardson P; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.
  • Sakata S; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.
  • Shaginian A; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.
  • Sonnenburg WK; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China.
  • Subramanyam C; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China.
  • Timofeevski S; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.
  • Wan J; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.
  • Yan W; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China.
  • Stewart AE; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.
ACS Med Chem Lett ; 11(6): 1175-1184, 2020 Jun 11.
Article em En | MEDLINE | ID: mdl-32550998

Texto completo: 1 Base de dados: MEDLINE Idioma: En Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Idioma: En Ano de publicação: 2020 Tipo de documento: Article