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Preclinical characterization of itacitinib (INCB039110), a novel selective inhibitor of JAK1, for the treatment of inflammatory diseases.
Covington, Maryanne; He, Xin; Scuron, Monika; Li, Jun; Collins, Robert; Juvekar, Ashish; Shin, Niu; Favata, Margaret; Gallagher, Karen; Sarah, Sarala; Xue, Chu-Biao; Peel, Michael; Burke, Krista; Oliver, Julian; Fay, Brittany; Yao, Wenqing; Huang, Taisheng; Scherle, Peggy; Diamond, Sharon; Newton, Robert; Zhang, Yan; Smith, Paul.
Afiliação
  • Covington M; Incyte Corporation, Wilmington, DE, USA.
  • He X; Incyte Corporation, Wilmington, DE, USA.
  • Scuron M; Incyte Corporation, Wilmington, DE, USA.
  • Li J; Incyte Corporation, Wilmington, DE, USA.
  • Collins R; Incyte Corporation, Wilmington, DE, USA.
  • Juvekar A; Incyte Corporation, Wilmington, DE, USA.
  • Shin N; Incyte Corporation, Wilmington, DE, USA.
  • Favata M; Incyte Corporation, Wilmington, DE, USA.
  • Gallagher K; Incyte Corporation, Wilmington, DE, USA.
  • Sarah S; Taconic Biosciences Incorporated, Rensselaer, NY, USA.
  • Xue CB; Incyte Corporation, Wilmington, DE, USA.
  • Peel M; Incyte Corporation, Wilmington, DE, USA.
  • Burke K; Incyte Corporation, Wilmington, DE, USA.
  • Oliver J; Incyte Corporation, Wilmington, DE, USA.
  • Fay B; Incyte Corporation, Wilmington, DE, USA.
  • Yao W; Incyte Corporation, Wilmington, DE, USA.
  • Huang T; Incyte Corporation, Wilmington, DE, USA.
  • Scherle P; Incyte Corporation, Wilmington, DE, USA.
  • Diamond S; Incyte Corporation, Wilmington, DE, USA.
  • Newton R; Incyte Corporation, Wilmington, DE, USA.
  • Zhang Y; Incyte Corporation, Wilmington, DE, USA.
  • Smith P; Incyte Corporation, Wilmington, DE, USA. Electronic address: psmith@incyte.com.
Eur J Pharmacol ; 885: 173505, 2020 Oct 15.
Article em En | MEDLINE | ID: mdl-32861662

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Azetidinas / Janus Quinase 1 / Inflamação / Ácidos Isonicotínicos Tipo de estudo: Prognostic_studies Limite: Animals / Humans Idioma: En Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Azetidinas / Janus Quinase 1 / Inflamação / Ácidos Isonicotínicos Tipo de estudo: Prognostic_studies Limite: Animals / Humans Idioma: En Ano de publicação: 2020 Tipo de documento: Article