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5-HT1A targeting PARCEST agent DO3AM-MPP with potential for receptor imaging: Synthesis, physico-chemical and MR studies.
Chaturvedi, Shubhra; Chaudhary, Vishakha; Pant, Pradeep; Jha, Preeti; Kumaran, Senthil S; Hussain, Firasat; Kumar Mishra, Anil.
Afiliação
  • Anju; Department of Chemistry, University of Delhi, North Campus, Delhi 110007, India; Division of Cyclotron and Radiopharmaceutical Sciences, Institute of Nuclear Medicine and Allied Sciences, Defence Research and Development Organization, Brig. S. K Mazumdar Road, Timarpur, Delhi 110054, India.
  • Chaturvedi S; Division of Cyclotron and Radiopharmaceutical Sciences, Institute of Nuclear Medicine and Allied Sciences, Defence Research and Development Organization, Brig. S. K Mazumdar Road, Timarpur, Delhi 110054, India. Electronic address: shubhra@inmas.drdo.in.
  • Chaudhary V; Department of Chemistry, University of Delhi, North Campus, Delhi 110007, India; Division of Cyclotron and Radiopharmaceutical Sciences, Institute of Nuclear Medicine and Allied Sciences, Defence Research and Development Organization, Brig. S. K Mazumdar Road, Timarpur, Delhi 110054, India.
  • Pant P; Department of Chemistry, Indian Institute of Technology, Hauz Khas, New Delhi 110016, India.
  • Jha P; Department of Immunology, Genetics and Pathology, Uppsala University, 75185 Uppsala, Sweden.
  • Kumaran SS; All India Institute of Medical Sciences, Ansari Nagar, New Delhi 110029, India.
  • Hussain F; Department of Chemistry, University of Delhi, North Campus, Delhi 110007, India.
  • Kumar Mishra A; Division of Cyclotron and Radiopharmaceutical Sciences, Institute of Nuclear Medicine and Allied Sciences, Defence Research and Development Organization, Brig. S. K Mazumdar Road, Timarpur, Delhi 110054, India. Electronic address: akmishra@inmas.drdo.in.
Bioorg Chem ; 106: 104487, 2021 01.
Article em En | MEDLINE | ID: mdl-33339667

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Propiofenonas / Imageamento por Ressonância Magnética / Meios de Contraste / Receptor 5-HT1A de Serotonina / Antagonistas do Receptor 5-HT1 de Serotonina Limite: Humans Idioma: En Ano de publicação: 2021 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Propiofenonas / Imageamento por Ressonância Magnética / Meios de Contraste / Receptor 5-HT1A de Serotonina / Antagonistas do Receptor 5-HT1 de Serotonina Limite: Humans Idioma: En Ano de publicação: 2021 Tipo de documento: Article