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Synthesis and evaluation of tiaprofenic acid-derived UCHL5 deubiquitinase inhibitors.
Gurusingha Arachchige, Harshani S; Herath Mudiyanselage, Poornima D H; VanHecke, Garrett C; Patel, Kush; Cheaito, Hassan A; Dou, Q Ping; Ahn, Young-Hoon.
Afiliação
  • Gurusingha Arachchige HS; Department of Chemistry, Wayne State University, Detroit, MI, USA.
  • Herath Mudiyanselage PDH; Department of Chemistry, Wayne State University, Detroit, MI, USA.
  • VanHecke GC; Department of Chemistry, Wayne State University, Detroit, MI, USA.
  • Patel K; Barbara Ann Karmanos Cancer Institute, Departments of Oncology, Pharmacology and Pathology, School of Medicine, Wayne State University, Detroit, MI, USA.
  • Cheaito HA; Barbara Ann Karmanos Cancer Institute, Departments of Oncology, Pharmacology and Pathology, School of Medicine, Wayne State University, Detroit, MI, USA.
  • Dou QP; Barbara Ann Karmanos Cancer Institute, Departments of Oncology, Pharmacology and Pathology, School of Medicine, Wayne State University, Detroit, MI, USA.
  • Ahn YH; Department of Chemistry, Wayne State University, Detroit, MI, USA. Electronic address: yahn@chem.wayne.edu.
Bioorg Med Chem ; 30: 115931, 2021 01 15.
Article em En | MEDLINE | ID: mdl-33341501

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Propionatos / Ubiquitina Tiolesterase / Inibidores Enzimáticos Limite: Humans Idioma: En Ano de publicação: 2021 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Propionatos / Ubiquitina Tiolesterase / Inibidores Enzimáticos Limite: Humans Idioma: En Ano de publicação: 2021 Tipo de documento: Article