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Variously substituted 2-oxopyridine derivatives: Extending the structure-activity relationships for allosteric modulation of the cannabinoid CB2 receptor.
Gado, Francesca; Mohamed, Kawthar A; Meini, Serena; Ferrisi, Rebecca; Bertini, Simone; Digiacomo, Maria; D'Andrea, Felicia; Stevenson, Lesley A; Laprairie, Robert B; Pertwee, Roger G; Manera, Clementina.
Afiliação
  • Gado F; Department of Pharmacy, University of Pisa, 56126, Pisa, Italy.
  • Mohamed KA; College of Pharmacy and Nutrition, University of Saskatchewan, Saskatoon, SK, Canada.
  • Meini S; Department of Pharmacy, University of Pisa, 56126, Pisa, Italy.
  • Ferrisi R; Department of Pharmacy, University of Pisa, 56126, Pisa, Italy.
  • Bertini S; Department of Pharmacy, University of Pisa, 56126, Pisa, Italy.
  • Digiacomo M; Department of Pharmacy, University of Pisa, 56126, Pisa, Italy.
  • D'Andrea F; Department of Pharmacy, University of Pisa, 56126, Pisa, Italy.
  • Stevenson LA; School of Medicine, Medical Sciences and Nutrition, Institute of Medical Sciences, University of Aberdeen, AB25 2ZD, Aberdeen, Scotland, UK.
  • Laprairie RB; College of Pharmacy and Nutrition, University of Saskatchewan, Saskatoon, SK, Canada.
  • Pertwee RG; School of Medicine, Medical Sciences and Nutrition, Institute of Medical Sciences, University of Aberdeen, AB25 2ZD, Aberdeen, Scotland, UK.
  • Manera C; Department of Pharmacy, University of Pisa, 56126, Pisa, Italy. Electronic address: clementina.manera@unipi.it.
Eur J Med Chem ; 211: 113116, 2021 Feb 05.
Article em En | MEDLINE | ID: mdl-33360803

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Receptor CB2 de Canabinoide / Regulação Alostérica Limite: Humans Idioma: En Ano de publicação: 2021 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Receptor CB2 de Canabinoide / Regulação Alostérica Limite: Humans Idioma: En Ano de publicação: 2021 Tipo de documento: Article