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Pseudo-Dipeptide Bearing α,α-Difluoromethyl Ketone Moiety as Electrophilic Warhead with Activity against Coronaviruses.
Citarella, Andrea; Gentile, Davide; Rescifina, Antonio; Piperno, Anna; Mognetti, Barbara; Gribaudo, Giorgio; Sciortino, Maria Teresa; Holzer, Wolfgang; Pace, Vittorio; Micale, Nicola.
Afiliação
  • Citarella A; Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina, V.le F. Stagno d'Alcontres 31, 98166 Messina, Italy.
  • Gentile D; Department of Pharmaceutical Chemistry, University of Vienna, Althanstrasse 14, A-1090 Vienna, Austria.
  • Rescifina A; Department of Drug Sciences, University of Catania, V.le A. Doria, 95125 Catania, Italy.
  • Piperno A; Department of Drug Sciences, University of Catania, V.le A. Doria, 95125 Catania, Italy.
  • Mognetti B; Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina, V.le F. Stagno d'Alcontres 31, 98166 Messina, Italy.
  • Gribaudo G; Department of Life Sciences and Systems Biology, University of Torino, Via Accademia Albertina 13, 10123 Torino, Italy.
  • Sciortino MT; Department of Life Sciences and Systems Biology, University of Torino, Via Accademia Albertina 13, 10123 Torino, Italy.
  • Holzer W; Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina, V.le F. Stagno d'Alcontres 31, 98166 Messina, Italy.
  • Pace V; Department of Pharmaceutical Chemistry, University of Vienna, Althanstrasse 14, A-1090 Vienna, Austria.
  • Micale N; Department of Pharmaceutical Chemistry, University of Vienna, Althanstrasse 14, A-1090 Vienna, Austria.
Int J Mol Sci ; 22(3)2021 Jan 30.
Article em En | MEDLINE | ID: mdl-33573283

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Antivirais / Coronavirus Humano 229E / Dipeptídeos / Cetonas Limite: Humans Idioma: En Ano de publicação: 2021 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Antivirais / Coronavirus Humano 229E / Dipeptídeos / Cetonas Limite: Humans Idioma: En Ano de publicação: 2021 Tipo de documento: Article