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Structure-based identification of dual ligands at the A2AR and PDE10A with anti-proliferative effects in lung cancer cell-lines.
Kalash, Leen; Winfield, Ian; Safitri, Dewi; Bermudez, Marcel; Carvalho, Sabrina; Glen, Robert; Ladds, Graham; Bender, Andreas.
Afiliação
  • Kalash L; Centre for Molecular Informatics, Department of Chemistry, University of Cambridge, Lensfield Road, CB21EW, Cambridge, UK.
  • Winfield I; GlaxoSmithKline, Gunnels Wood Road, Hertfordshire, SG1 2NY, Stevenage, UK.
  • Safitri D; Centre for Molecular Informatics, Department of Chemistry, University of Cambridge, Lensfield Road, CB21EW, Cambridge, UK.
  • Bermudez M; Department of Pharmacology, University of Cambridge, Tennis Court Road, CB2 1PD, Cambridge, UK.
  • Carvalho S; Department of Pharmacology, University of Cambridge, Tennis Court Road, CB2 1PD, Cambridge, UK.
  • Glen R; Pharmacology and Clinical Pharmacy Research Group, School of Pharmacy, Bandung Institute of Technology, 40132, Bandung, Indonesia.
  • Ladds G; Centre for Molecular Informatics, Department of Chemistry, University of Cambridge, Lensfield Road, CB21EW, Cambridge, UK.
  • Bender A; Institute of Pharmacy, Freie Universität Berlin, Königin-Luise-Straße 2 und 4, 14195, Berlin, Germany.
J Cheminform ; 13(1): 17, 2021 Mar 03.
Article em En | MEDLINE | ID: mdl-33658076

Texto completo: 1 Base de dados: MEDLINE Tipo de estudo: Diagnostic_studies / Prognostic_studies Idioma: En Ano de publicação: 2021 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Tipo de estudo: Diagnostic_studies / Prognostic_studies Idioma: En Ano de publicação: 2021 Tipo de documento: Article