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A novel class of selective non-nucleoside inhibitors of human DNA methyltransferase 3A.
Huang, Sunzeyu; Stillson, Nathaniel J; Sandoval, Jonathan E; Yung, Chitoh; Reich, Norbert O.
Afiliação
  • Huang S; The Department of Chemistry and Biochemistry, University of California, Santa Barbara 93106-9510, USA.
  • Stillson NJ; The Department of Chemistry and Biochemistry, University of California, Santa Barbara 93106-9510, USA.
  • Sandoval JE; The Department of Chemistry and Biochemistry, University of California, Santa Barbara 93106-9510, USA; Molecular, Cellular and Developmental Biology, University of California, Santa Barbara 93106-9510, USA.
  • Yung C; The Department of Chemistry and Biochemistry, University of California, Santa Barbara 93106-9510, USA.
  • Reich NO; The Department of Chemistry and Biochemistry, University of California, Santa Barbara 93106-9510, USA. Electronic address: reich@chem.ucsb.edu.
Bioorg Med Chem Lett ; 40: 127908, 2021 05 15.
Article em En | MEDLINE | ID: mdl-33705897

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Piridazinas / Pirazolonas / DNA (Citosina-5-)-Metiltransferases / Inibidores Enzimáticos / Bibliotecas de Moléculas Pequenas Limite: Humans Idioma: En Ano de publicação: 2021 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Piridazinas / Pirazolonas / DNA (Citosina-5-)-Metiltransferases / Inibidores Enzimáticos / Bibliotecas de Moléculas Pequenas Limite: Humans Idioma: En Ano de publicação: 2021 Tipo de documento: Article