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Design, Synthesis, and Structural Characterization of Lysine Covalent BH3 Peptides Targeting Mcl-1.
Gambini, Luca; Udompholkul, Parima; Baggio, Carlo; Muralidharan, Aruljothi; Kenjic, Nikola; Assar, Zahra; Perry, J Jefferson P; Pellecchia, Maurizio.
Afiliação
  • Gambini L; Division of Biomedical Sciences, School of Medicine, University of California Riverside, 900 University Avenue, Riverside, California 92521, United States.
  • Udompholkul P; Division of Biomedical Sciences, School of Medicine, University of California Riverside, 900 University Avenue, Riverside, California 92521, United States.
  • Baggio C; Division of Biomedical Sciences, School of Medicine, University of California Riverside, 900 University Avenue, Riverside, California 92521, United States.
  • Muralidharan A; Division of Biomedical Sciences, School of Medicine, University of California Riverside, 900 University Avenue, Riverside, California 92521, United States.
  • Kenjic N; Department of Biochemistry, College of Natural and Agricultural Sciences, University of California Riverside, 900 University Avenue, Riverside, California 92521, United States.
  • Assar Z; Cayman Chemical, 1180 East Ellsworth Road, Ann Arbor, Michigan 48108, United States.
  • Perry JJP; Department of Biochemistry, College of Natural and Agricultural Sciences, University of California Riverside, 900 University Avenue, Riverside, California 92521, United States.
  • Pellecchia M; Division of Biomedical Sciences, School of Medicine, University of California Riverside, 900 University Avenue, Riverside, California 92521, United States.
J Med Chem ; 64(8): 4903-4912, 2021 04 22.
Article em En | MEDLINE | ID: mdl-33797903

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Fragmentos de Peptídeos / Desenho de Fármacos / Proteínas Proto-Oncogênicas / Proteína de Sequência 1 de Leucemia de Células Mieloides / Lisina Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Ano de publicação: 2021 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Fragmentos de Peptídeos / Desenho de Fármacos / Proteínas Proto-Oncogênicas / Proteína de Sequência 1 de Leucemia de Células Mieloides / Lisina Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Ano de publicação: 2021 Tipo de documento: Article