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Dihydropyridine Lactam Analogs Targeting BET Bromodomains.
Jiang, Jiewei; Sigua, Logan H; Chan, Alice; Kalra, Prakriti; Pomerantz, William C K; Schönbrunn, Ernst; Qi, Jun; Georg, Gunda I.
Afiliação
  • Jiang J; Department of Medicinal Chemistry and Institute for Therapeutics Discovery and Development, College of Pharmacy, University of Minnesota, 717 Delaware Street SE, Minneapolis, MN 55414, USA.
  • Sigua LH; Department of Cancer Biology, Dana-Farber Cancer Institute, Boston, MA 02215, USA.
  • Chan A; Moffitt Cancer Center, Drug Discovery Department, 12902 Magnolia Drive, Tampa, Fl 33612, USA.
  • Kalra P; Department of Chemistry, University of Minnesota, 207 Pleasant Street SE, Minneapolis, MN 55455, USA.
  • Pomerantz WCK; Department of Chemistry, University of Minnesota, 207 Pleasant Street SE, Minneapolis, MN 55455, USA.
  • Schönbrunn E; Moffitt Cancer Center, Drug Discovery Department, 12902 Magnolia Drive, Tampa, Fl 33612, USA.
  • Qi J; Department of Cancer Biology, Dana-Farber Cancer Institute, Boston, MA 02215, USA.
  • Georg GI; Department of Medicine, Harvard Medical School, Boston, MA 02115, USA.
ChemMedChem ; 17(1): e202100407, 2022 01 05.
Article em En | MEDLINE | ID: mdl-34932262

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Di-Hidropiridinas / Proteínas Nucleares / Lactamas Limite: Humans Idioma: En Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Di-Hidropiridinas / Proteínas Nucleares / Lactamas Limite: Humans Idioma: En Ano de publicação: 2022 Tipo de documento: Article