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Synthesis of tropane-based σ1 receptor antagonists with antiallodynic activity.
Bechthold, Elena; Schreiber, Julian A; Ritter, Nadine; Grey, Lucie; Schepmann, Dirk; Daniliuc, Constantin; González-Cano, Rafael; Nieto, Francisco Rafael; Seebohm, Guiscard; Wünsch, Bernhard.
Afiliação
  • Bechthold E; GRK 2515, Chemical Biology of Ion Channels (Chembion), Westfälische Wilhelms-Universität Münster, Germany; Institut für Pharmazeutische und Medizinische Chemie, Westfälische Wilhelms-Universität Münster, Corrensstraße 48, D-48149, Münster, Germany.
  • Schreiber JA; Institut für Pharmazeutische und Medizinische Chemie, Westfälische Wilhelms-Universität Münster, Corrensstraße 48, D-48149, Münster, Germany; Cellular Electrophysiology and Molecular Biology, Institute for Genetics of Heart Diseases (IfGH), Department of Cardiovascular Medicine, University Hospital
  • Ritter N; GRK 2515, Chemical Biology of Ion Channels (Chembion), Westfälische Wilhelms-Universität Münster, Germany; Cellular Electrophysiology and Molecular Biology, Institute for Genetics of Heart Diseases (IfGH), Department of Cardiovascular Medicine, University Hospital Münster, Robert-Koch-Str. 45, D-481
  • Grey L; Institut für Pharmazeutische und Medizinische Chemie, Westfälische Wilhelms-Universität Münster, Corrensstraße 48, D-48149, Münster, Germany.
  • Schepmann D; Institut für Pharmazeutische und Medizinische Chemie, Westfälische Wilhelms-Universität Münster, Corrensstraße 48, D-48149, Münster, Germany.
  • Daniliuc C; Organisch-chemisches Institut, Westfälische Wilhelms-Universität Münster, Corrensstraße 40, D-48149, Münster, Germany.
  • González-Cano R; Department of Pharmacology and Institute of Neuroscience, School of Medicine and Biomedical Research Center, University of Granada, Avenida de la Investigación 11, 18016, Granada, Spain; Biosanitary Research Institute ibs.GRANADA, 18012, Granada, Spain.
  • Nieto FR; Department of Pharmacology and Institute of Neuroscience, School of Medicine and Biomedical Research Center, University of Granada, Avenida de la Investigación 11, 18016, Granada, Spain; Biosanitary Research Institute ibs.GRANADA, 18012, Granada, Spain.
  • Seebohm G; GRK 2515, Chemical Biology of Ion Channels (Chembion), Westfälische Wilhelms-Universität Münster, Germany; Cellular Electrophysiology and Molecular Biology, Institute for Genetics of Heart Diseases (IfGH), Department of Cardiovascular Medicine, University Hospital Münster, Robert-Koch-Str. 45, D-481
  • Wünsch B; GRK 2515, Chemical Biology of Ion Channels (Chembion), Westfälische Wilhelms-Universität Münster, Germany; Institut für Pharmazeutische und Medizinische Chemie, Westfälische Wilhelms-Universität Münster, Corrensstraße 48, D-48149, Münster, Germany. Electronic address: wuensch@uni-muenster.de.
Eur J Med Chem ; 230: 114113, 2022 Feb 15.
Article em En | MEDLINE | ID: mdl-35065412

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Receptores sigma Idioma: En Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Receptores sigma Idioma: En Ano de publicação: 2022 Tipo de documento: Article