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In vitro pharmacological profile of PHA-022121, a small molecule bradykinin B2 receptor antagonist in clinical development.
Lesage, Anne; Marceau, François; Gibson, Christoph; Loenders, Brigitte; Katzer, Werner; Ambrosi, Horst-Dieter; Saupe, Jörn; Faussner, Alexander; Pardali, Evangelia; Knolle, Jochen.
Afiliação
  • Lesage A; Pharvaris GmbH., Zug, Switzerland. Electronic address: anne.lesage@pharvaris.com.
  • Marceau F; Département de Microbiologie, Infectiologie et Immunologie, Faculté de médecine, Université Laval, Québec, QC G1V 4G2, Canada.
  • Gibson C; AnalytiCon Discovery GmbH, Potsdam, Germany.
  • Loenders B; Pharvaris Netherlands B.V., Leiden, the Netherlands.
  • Katzer W; AnalytiCon Discovery GmbH, Potsdam, Germany.
  • Ambrosi HD; AnalytiCon Discovery GmbH, Potsdam, Germany.
  • Saupe J; AnalytiCon Discovery GmbH, Potsdam, Germany.
  • Faussner A; Faculty of Medicine, Institute for Cardiovascular Prevention, Ludwig-Maximilians-University, Munich, Germany.
  • Pardali E; Pharvaris Netherlands B.V., Leiden, the Netherlands.
  • Knolle J; Pharvaris GmbH., Zug, Switzerland.
Int Immunopharmacol ; 105: 108523, 2022 Apr.
Article em En | MEDLINE | ID: mdl-35086057

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Bradicinina / Antagonistas dos Receptores da Bradicinina Limite: Animals Idioma: En Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Bradicinina / Antagonistas dos Receptores da Bradicinina Limite: Animals Idioma: En Ano de publicação: 2022 Tipo de documento: Article