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9-Cyclopropylmethoxy-dihydrotetrabenazine and its stereoisomers as vesicular monoamine transporter-2 inhibitors.
Wang, Wenyan; Lin, Shilan; Du, Guangying; Bai, Xinfa; Lu, Jing; Ye, Liang; Wang, Hongbo; Zhang, Rui; Tian, Jingwei.
Afiliação
  • Wang W; School of Pharmacy, Key Laboratory of Molecular Pharmacology & Drug Evaluation (Yantai University), Ministry of Education, Collaborative Innovation Center of Advanced Drug Delivery System & Biotech Drugs in Universities of Shandong, Yantai University, Yantai, 264005, China.
  • Lin S; School of Pharmacy, Key Laboratory of Molecular Pharmacology & Drug Evaluation (Yantai University), Ministry of Education, Collaborative Innovation Center of Advanced Drug Delivery System & Biotech Drugs in Universities of Shandong, Yantai University, Yantai, 264005, China.
  • Du G; School of Pharmacy, Key Laboratory of Molecular Pharmacology & Drug Evaluation (Yantai University), Ministry of Education, Collaborative Innovation Center of Advanced Drug Delivery System & Biotech Drugs in Universities of Shandong, Yantai University, Yantai, 264005, China.
  • Bai X; New Drug Discovery & Research Department, R & D Center (Luye Pharma Group Ltd), Yantai, 264003, China.
  • Lu J; School of Pharmacy, Key Laboratory of Molecular Pharmacology & Drug Evaluation (Yantai University), Ministry of Education, Collaborative Innovation Center of Advanced Drug Delivery System & Biotech Drugs in Universities of Shandong, Yantai University, Yantai, 264005, China.
  • Ye L; New Drug Discovery & Research Department, R & D Center (Luye Pharma Group Ltd), Yantai, 264003, China.
  • Wang H; School of Pharmacy, Key Laboratory of Molecular Pharmacology & Drug Evaluation (Yantai University), Ministry of Education, Collaborative Innovation Center of Advanced Drug Delivery System & Biotech Drugs in Universities of Shandong, Yantai University, Yantai, 264005, China.
  • Zhang R; New Drug Discovery & Research Department, R & D Center (Luye Pharma Group Ltd), Yantai, 264003, China.
  • Tian J; School of Pharmacy, Key Laboratory of Molecular Pharmacology & Drug Evaluation (Yantai University), Ministry of Education, Collaborative Innovation Center of Advanced Drug Delivery System & Biotech Drugs in Universities of Shandong, Yantai University, Yantai, 264005, China.
Future Med Chem ; 14(13): 991-1003, 2022 07.
Article em En | MEDLINE | ID: mdl-35638444

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Tetrabenazina / Proteínas Vesiculares de Transporte de Monoamina / Moduladores de Transporte de Membrana Limite: Animals Idioma: En Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Tetrabenazina / Proteínas Vesiculares de Transporte de Monoamina / Moduladores de Transporte de Membrana Limite: Animals Idioma: En Ano de publicação: 2022 Tipo de documento: Article