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Enzyme Responsive Rigid-Rod Aromatics Target "Undruggable" Phosphatases to Kill Cancer Cells in a Mimetic Bone Microenvironment.
Yi, Meihui; Wang, Fengbin; Tan, Weiyi; Hsieh, Jer-Tsong; Egelman, Edward H; Xu, Bing.
Afiliação
  • Yi M; Department of Chemistry, Brandeis University, 415 South Street, Waltham, Massachusetts 02453, United States.
  • Wang F; Department of Biochemistry and Molecular Genetics, University of Virginia, Charlottesville, Virginia 22908, United States.
  • Tan W; Department of Chemistry, Brandeis University, 415 South Street, Waltham, Massachusetts 02453, United States.
  • Hsieh JT; Department of Urology, Southwestern Medical Center, University of Texas, Dallas, Texas 75235, United States.
  • Egelman EH; Department of Biochemistry and Molecular Genetics, University of Virginia, Charlottesville, Virginia 22908, United States.
  • Xu B; Department of Chemistry, Brandeis University, 415 South Street, Waltham, Massachusetts 02453, United States.
J Am Chem Soc ; 144(29): 13055-13059, 2022 07 27.
Article em En | MEDLINE | ID: mdl-35849554

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Neoplasias da Próstata / Monoéster Fosfórico Hidrolases Limite: Humans / Male Idioma: En Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Neoplasias da Próstata / Monoéster Fosfórico Hidrolases Limite: Humans / Male Idioma: En Ano de publicação: 2022 Tipo de documento: Article