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SRI-32743, a novel allosteric modulator, attenuates HIV-1 Tat protein-induced inhibition of the dopamine transporter and alleviates the potentiation of cocaine reward in HIV-1 Tat transgenic mice.
Zhu, Jun; Quizon, Pamela M; Wang, Yingying; Adeniran, Charles A; Strauss, Matthew J; Jiménez-Torres, Ana C; Patel, Palak; Cirino, Thomas J; Eans, Shainnel O; Hammond, Haylee R; Deliscar, Laure S; O'Hara, Priscilla; Saini, Surendra K; Ofori, Edward; Vekariya, Rakesh H; Zhang, Sixue; Moukha-Chafiq, Omar; Nguyen, Theresa H; Ananthan, Subramaniam; Augelli-Szafran, Corinne E; Zhan, Chang-Guo; McLaughlin, Jay P.
Afiliação
  • Zhu J; Department of Drug Discovery and Biomedical Sciences, College of Pharmacy, University of South Carolina, Columbia, SC 29208, USA. Electronic address: zhuj@cop.sc.edu.
  • Quizon PM; Department of Drug Discovery and Biomedical Sciences, College of Pharmacy, University of South Carolina, Columbia, SC 29208, USA.
  • Wang Y; Department of Drug Discovery and Biomedical Sciences, College of Pharmacy, University of South Carolina, Columbia, SC 29208, USA.
  • Adeniran CA; Molecular Modeling and Biopharmaceutical Center, USA; Department of Pharmaceutical Sciences, College of Pharmacy, University of Kentucky, Lexington, KY 40536, USA.
  • Strauss MJ; Department of Drug Discovery and Biomedical Sciences, College of Pharmacy, University of South Carolina, Columbia, SC 29208, USA.
  • Jiménez-Torres AC; Department of Drug Discovery and Biomedical Sciences, College of Pharmacy, University of South Carolina, Columbia, SC 29208, USA.
  • Patel P; Department of Drug Discovery and Biomedical Sciences, College of Pharmacy, University of South Carolina, Columbia, SC 29208, USA.
  • Cirino TJ; Department of Pharmacodynamics, College of Pharmacy, University of Florida, Gainesville, FL 32611, USA.
  • Eans SO; Department of Pharmacodynamics, College of Pharmacy, University of Florida, Gainesville, FL 32611, USA.
  • Hammond HR; Department of Pharmacodynamics, College of Pharmacy, University of Florida, Gainesville, FL 32611, USA.
  • Deliscar LS; Department of Pharmacodynamics, College of Pharmacy, University of Florida, Gainesville, FL 32611, USA.
  • O'Hara P; Department of Pharmacodynamics, College of Pharmacy, University of Florida, Gainesville, FL 32611, USA.
  • Saini SK; Department of Chemistry, Scientific Platforms, Southern Research, Birmingham, AL 35205, USA.
  • Ofori E; Department of Chemistry, Scientific Platforms, Southern Research, Birmingham, AL 35205, USA.
  • Vekariya RH; Department of Chemistry, Scientific Platforms, Southern Research, Birmingham, AL 35205, USA.
  • Zhang S; Department of Chemistry, Scientific Platforms, Southern Research, Birmingham, AL 35205, USA.
  • Moukha-Chafiq O; Department of Chemistry, Scientific Platforms, Southern Research, Birmingham, AL 35205, USA.
  • Nguyen TH; Department of Chemistry, Scientific Platforms, Southern Research, Birmingham, AL 35205, USA.
  • Ananthan S; Department of Chemistry, Scientific Platforms, Southern Research, Birmingham, AL 35205, USA.
  • Augelli-Szafran CE; Department of Chemistry, Scientific Platforms, Southern Research, Birmingham, AL 35205, USA.
  • Zhan CG; Molecular Modeling and Biopharmaceutical Center, USA; Department of Pharmaceutical Sciences, College of Pharmacy, University of Kentucky, Lexington, KY 40536, USA.
  • McLaughlin JP; Department of Pharmacodynamics, College of Pharmacy, University of Florida, Gainesville, FL 32611, USA.
Neuropharmacology ; 220: 109239, 2022 Dec 01.
Article em En | MEDLINE | ID: mdl-36126727

Texto completo: 1 Base de dados: MEDLINE Assunto principal: HIV-1 / Cocaína / Transtornos Relacionados ao Uso de Cocaína Limite: Animals / Humans Idioma: En Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: HIV-1 / Cocaína / Transtornos Relacionados ao Uso de Cocaína Limite: Animals / Humans Idioma: En Ano de publicação: 2022 Tipo de documento: Article