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Essential role of P-glycoprotein in the mechanism of action of oliceridine.
Ventriglia, Emilya; Rizzo, Arianna; Gomez, Juan L; Friedman, Jacob; Lam, Sherry; Solís, Oscar; Rais, Rana; Bonaventura, Jordi; Michaelides, Michael.
Afiliação
  • Ventriglia E; Biobehavioral Imaging and Molecular Neuropsychopharmacology Unit, National Institute on Drug Abuse, Baltimore, MD, 21224, USA.
  • Rizzo A; Departament de Patologia i Terapèutica Experimental, Institute de Neurociències, Universitat de Barcelona, L'Hospitalet de Llobregat, Catalonia, Spain.
  • Gomez JL; Neuropharmacology & Pain Group, Neuroscience Program, Bellvitge Institute for Biomedical Research (IDIBELL), L'Hospitalet de Llobregat, Catalonia, Spain.
  • Friedman J; Biobehavioral Imaging and Molecular Neuropsychopharmacology Unit, National Institute on Drug Abuse, Baltimore, MD, 21224, USA.
  • Lam S; Medications Development Program, Molecular Targets and Medication Discovery Branch, National Institute on Drug Abuse, Baltimore, MD, 21224, USA.
  • Solís O; Johns Hopkins Drug Discovery, Johns Hopkins School of Medicine, Baltimore, MD, 21205, USA.
  • Rais R; Biobehavioral Imaging and Molecular Neuropsychopharmacology Unit, National Institute on Drug Abuse, Baltimore, MD, 21224, USA.
  • Bonaventura J; Biobehavioral Imaging and Molecular Neuropsychopharmacology Unit, National Institute on Drug Abuse, Baltimore, MD, 21224, USA.
  • Michaelides M; Johns Hopkins Drug Discovery, Johns Hopkins School of Medicine, Baltimore, MD, 21205, USA.
Neuropsychopharmacology ; 48(5): 831-842, 2023 04.
Article em En | MEDLINE | ID: mdl-36434081

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Membro 1 da Subfamília B de Cassetes de Ligação de ATP / Analgésicos Opioides Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Membro 1 da Subfamília B de Cassetes de Ligação de ATP / Analgésicos Opioides Idioma: En Ano de publicação: 2023 Tipo de documento: Article