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2-Anilino-4-(1-methyl-1H-pyrazol-4-yl)pyrimidine-derived CDK2 inhibitors as anticancer agents: Design, synthesis & evaluation.
Fanta, Biruk Sintayehu; Mekonnen, Laychiluh; Basnet, Sunita K C; Teo, Theodosia; Lenjisa, Jimma; Khair, Nishat Z; Kou, Lianmeng; Tadesse, Solomon; Sykes, Matthew J; Yu, Mingfeng; Wang, Shudong.
Afiliação
  • Fanta BS; Drug Discovery and Development, Clinical and Health Sciences, University of South Australia, Adelaide, South Australia 5000, Australia.
  • Mekonnen L; Drug Discovery and Development, Clinical and Health Sciences, University of South Australia, Adelaide, South Australia 5000, Australia.
  • Basnet SKC; Drug Discovery and Development, Clinical and Health Sciences, University of South Australia, Adelaide, South Australia 5000, Australia.
  • Teo T; Drug Discovery and Development, Clinical and Health Sciences, University of South Australia, Adelaide, South Australia 5000, Australia.
  • Lenjisa J; Drug Discovery and Development, Clinical and Health Sciences, University of South Australia, Adelaide, South Australia 5000, Australia.
  • Khair NZ; Drug Discovery and Development, Clinical and Health Sciences, University of South Australia, Adelaide, South Australia 5000, Australia.
  • Kou L; Drug Discovery and Development, Clinical and Health Sciences, University of South Australia, Adelaide, South Australia 5000, Australia.
  • Tadesse S; Drug Discovery and Development, Clinical and Health Sciences, University of South Australia, Adelaide, South Australia 5000, Australia.
  • Sykes MJ; Drug Discovery and Development, Clinical and Health Sciences, University of South Australia, Adelaide, South Australia 5000, Australia.
  • Yu M; Drug Discovery and Development, Clinical and Health Sciences, University of South Australia, Adelaide, South Australia 5000, Australia. Electronic address: Mingfeng.Yu@unisa.edu.au.
  • Wang S; Drug Discovery and Development, Clinical and Health Sciences, University of South Australia, Adelaide, South Australia 5000, Australia. Electronic address: Shudong.Wang@unisa.edu.au.
Bioorg Med Chem ; 80: 117158, 2023 02 15.
Article em En | MEDLINE | ID: mdl-36706608

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Neoplasias / Antineoplásicos Limite: Humans Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Neoplasias / Antineoplásicos Limite: Humans Idioma: En Ano de publicação: 2023 Tipo de documento: Article