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Structure-guided optimization of adenosine mimetics as selective and potent inhibitors of coronavirus nsp14 N7-methyltransferases.
Hausdorff, Marcel; Delpal, Adrien; Barelier, Sarah; Nicollet, Laura; Canard, Bruno; Touret, Franck; Colmant, Agathe; Coutard, Bruno; Vasseur, Jean-Jacques; Decroly, Etienne; Debart, Françoise.
Afiliação
  • Hausdorff M; IBMM, CNRS, University of Montpellier, ENSCM, Montpellier, France.
  • Delpal A; AFMB, CNRS, Aix-Marseille University, UMR 7257, 163 Avenue de Luminy, Marseille, France.
  • Barelier S; AFMB, CNRS, Aix-Marseille University, UMR 7257, 163 Avenue de Luminy, Marseille, France.
  • Nicollet L; IBMM, CNRS, University of Montpellier, ENSCM, Montpellier, France.
  • Canard B; AFMB, CNRS, Aix-Marseille University, UMR 7257, 163 Avenue de Luminy, Marseille, France.
  • Touret F; IHU Méditerranée Infection, Unité Virus Emergents, University of Aix-Marseille, 13005, Marseille, France.
  • Colmant A; IHU Méditerranée Infection, Unité Virus Emergents, University of Aix-Marseille, 13005, Marseille, France.
  • Coutard B; IHU Méditerranée Infection, Unité Virus Emergents, University of Aix-Marseille, 13005, Marseille, France.
  • Vasseur JJ; IBMM, CNRS, University of Montpellier, ENSCM, Montpellier, France.
  • Decroly E; AFMB, CNRS, Aix-Marseille University, UMR 7257, 163 Avenue de Luminy, Marseille, France. Electronic address: etienne.decroly@univ-amu.fr.
  • Debart F; IBMM, CNRS, University of Montpellier, ENSCM, Montpellier, France. Electronic address: francoise.debart@umontpellier.fr.
Eur J Med Chem ; 256: 115474, 2023 Aug 05.
Article em En | MEDLINE | ID: mdl-37192550

Texto completo: 1 Base de dados: MEDLINE Assunto principal: COVID-19 / Metiltransferases Limite: Humans Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: COVID-19 / Metiltransferases Limite: Humans Idioma: En Ano de publicação: 2023 Tipo de documento: Article