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Design, Synthesis, and Pharmacological Characterization of a Potent Soluble Epoxide Hydrolase Inhibitor for the Treatment of Acute Pancreatitis.
Musella, Simona; D'Avino, Danilo; Peltner, Lukas Klaus; Di Sarno, Veronica; Cerqua, Ida; Merciai, Fabrizio; Vestuto, Vincenzo; Ciaglia, Tania; Smaldone, Gerardina; Di Matteo, Francesca; Di Micco, Simone; Napolitano, Valeria; Bifulco, Giuseppe; Pepe, Giacomo; Sommella, Eduardo Maria; Basilicata, Manuela Giovanna; Aquino, Giovanna; Gomez-Monterrey, Isabel M; Campiglia, Pietro; Ostacolo, Carmine; Roviezzo, Fiorentina; Werz, Oliver; Rossi, Antonietta; Bertamino, Alessia.
Afiliação
  • Musella S; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • D'Avino D; Department of Pharmacy, University Federico II of Naples, Via D. Montesano 49, 80131 Naples, Italy.
  • Peltner LK; Department of Pharmaceutical/Medicinal Chemistry, Institute of Pharmacy, Friedrich-Schiller-University, Philosophenweg 14, D-07743 Jena, Germany.
  • Di Sarno V; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Cerqua I; Department of Pharmacy, University Federico II of Naples, Via D. Montesano 49, 80131 Naples, Italy.
  • Merciai F; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Vestuto V; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Ciaglia T; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Smaldone G; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Di Matteo F; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Di Micco S; European Biomedical Research Institute (EBRIS), Via S. De Renzi 50, 84125 Salerno, Italy.
  • Napolitano V; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Bifulco G; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Pepe G; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Sommella EM; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Basilicata MG; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Aquino G; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Gomez-Monterrey IM; PhD Program in Drug Discovery and Development, University of Salerno, 84084 Fisciano, SA, Italy.
  • Campiglia P; Department of Pharmacy, University Federico II of Naples, Via D. Montesano 49, 80131 Naples, Italy.
  • Ostacolo C; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Roviezzo F; European Biomedical Research Institute (EBRIS), Via S. De Renzi 50, 84125 Salerno, Italy.
  • Werz O; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Rossi A; Department of Pharmacy, University Federico II of Naples, Via D. Montesano 49, 80131 Naples, Italy.
  • Bertamino A; Department of Pharmaceutical/Medicinal Chemistry, Institute of Pharmacy, Friedrich-Schiller-University, Philosophenweg 14, D-07743 Jena, Germany.
J Med Chem ; 66(13): 9201-9222, 2023 07 13.
Article em En | MEDLINE | ID: mdl-37334504

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Pancreatite Limite: Animals Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Pancreatite Limite: Animals Idioma: En Ano de publicação: 2023 Tipo de documento: Article