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Targeting the Alternative Vitamin E Metabolite Binding Site Enables Noncanonical PPARγ Modulation.
Arifi, Silvia; Marschner, Julian A; Pollinger, Julius; Isigkeit, Laura; Heitel, Pascal; Kaiser, Astrid; Obeser, Lennart; Höfner, Georg; Proschak, Ewgenij; Knapp, Stefan; Chaikuad, Apirat; Heering, Jan; Merk, Daniel.
Afiliação
  • Arifi S; Institute of Pharmaceutical Chemistry, Goethe University Frankfurt, D-60438 Frankfurt, Germany.
  • Marschner JA; Department of Pharmacy, Ludwig-Maximilians-Universität München, D-81377 Munich, Germany.
  • Pollinger J; Institute of Pharmaceutical Chemistry, Goethe University Frankfurt, D-60438 Frankfurt, Germany.
  • Isigkeit L; Institute of Pharmaceutical Chemistry, Goethe University Frankfurt, D-60438 Frankfurt, Germany.
  • Heitel P; Institute of Pharmaceutical Chemistry, Goethe University Frankfurt, D-60438 Frankfurt, Germany.
  • Kaiser A; Institute of Pharmaceutical Chemistry, Goethe University Frankfurt, D-60438 Frankfurt, Germany.
  • Obeser L; Department of Pharmacy, Ludwig-Maximilians-Universität München, D-81377 Munich, Germany.
  • Höfner G; Department of Pharmacy, Ludwig-Maximilians-Universität München, D-81377 Munich, Germany.
  • Proschak E; Institute of Pharmaceutical Chemistry, Goethe University Frankfurt, D-60438 Frankfurt, Germany.
  • Knapp S; Fraunhofer Institute for Translational Medicine and Pharmacology ITMP, D-60596 Frankfurt, Germany.
  • Chaikuad A; Institute of Pharmaceutical Chemistry, Goethe University Frankfurt, D-60438 Frankfurt, Germany.
  • Heering J; Structural Genomics Consortium, BMLS, Goethe University Frankfurt, D-60438 Frankfurt, Germany.
  • Merk D; Institute of Pharmaceutical Chemistry, Goethe University Frankfurt, D-60438 Frankfurt, Germany.
J Am Chem Soc ; 145(27): 14802-14810, 2023 07 12.
Article em En | MEDLINE | ID: mdl-37385602

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Tiazolidinedionas / PPAR gama Tipo de estudo: Prognostic_studies Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Tiazolidinedionas / PPAR gama Tipo de estudo: Prognostic_studies Idioma: En Ano de publicação: 2023 Tipo de documento: Article