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Synthesis and anti-cancer potential of potent peripheral MAOA inhibitors designed to limit blood:brain penetration.
Jacobs, Michaela R; Olivero, Jennifer E; Ok Choi, Hyun; Liao, Chun-Peng; Kashemirov, Boris A; Katz, Jonathan E; Gross, Mitchell E; McKenna, Charles E.
Afiliação
  • Jacobs MR; Department of Chemistry, University of Southern California, Los Angeles, CA 90089, USA. Electronic address: jacobsmr@usc.edu.
  • Olivero JE; Department of Chemistry, University of Southern California, Los Angeles, CA 90089, USA. Electronic address: jeoliver@usc.edu.
  • Ok Choi H; Lawrence J. Ellison Institute for Transformative Medicine, Los Angeles, CA 90064, USA. Electronic address: hchoi@eitm.org.
  • Liao CP; Lawrence J. Ellison Institute for Transformative Medicine, Los Angeles, CA 90064, USA. Electronic address: cliao@eitm.org.
  • Kashemirov BA; Department of Chemistry, University of Southern California, Los Angeles, CA 90089, USA. Electronic address: kashemir@usc.edu.
  • Katz JE; Lawrence J. Ellison Institute for Transformative Medicine, Los Angeles, CA 90064, USA; Department of Medicine, Keck School of Medicine, University of Southern California, Los Angeles, CA 90033, USA. Electronic address: jonathan@eitm.org.
  • Gross ME; Lawrence J. Ellison Institute for Transformative Medicine, Los Angeles, CA 90064, USA; Department of Medicine, Keck School of Medicine, University of Southern California, Los Angeles, CA 90033, USA. Electronic address: mgross@eitm.org.
  • McKenna CE; Department of Chemistry, University of Southern California, Los Angeles, CA 90089, USA. Electronic address: mckenna@usc.edu.
Bioorg Med Chem ; 92: 117425, 2023 09 07.
Article em En | MEDLINE | ID: mdl-37544256

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Neoplasias da Próstata / Inibidores da Monoaminoxidase Tipo de estudo: Prognostic_studies Limite: Humans / Male Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Neoplasias da Próstata / Inibidores da Monoaminoxidase Tipo de estudo: Prognostic_studies Limite: Humans / Male Idioma: En Ano de publicação: 2023 Tipo de documento: Article