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Assembling a Cinnamyl Pharmacophore in the C3-Position of Substituted Isatins via Microwave-Assisted Synthesis: Development of a New Class of Monoamine Oxidase-B Inhibitors for the Treatment of Parkinson's Disease.
Manoharan, Amritha; Oh, Jong Min; Benny, Feba; Kumar, Sunil; Abdelgawad, Mohamed A; Ghoneim, Mohammed M; Shaker, Mohamed E; El-Sherbiny, Mohamed; Almohaimeed, Hailah M; Gahtori, Prashant; Kim, Hoon; Mathew, Bijo.
Afiliação
  • Manoharan A; Department of Pharmaceutical Chemistry, Amrita School of Pharmacy, Amrita Vishwa Vidyapeetham, AIMS Health Sciences Campus, Kochi 682 041, India.
  • Oh JM; Department of Pharmacy, Research Institute of Life Pharmaceutical Sciences, Sunchon National University, Suncheon 57922, Republic of Korea.
  • Benny F; Department of Pharmaceutical Chemistry, Amrita School of Pharmacy, Amrita Vishwa Vidyapeetham, AIMS Health Sciences Campus, Kochi 682 041, India.
  • Kumar S; Department of Pharmaceutical Chemistry, Amrita School of Pharmacy, Amrita Vishwa Vidyapeetham, AIMS Health Sciences Campus, Kochi 682 041, India.
  • Abdelgawad MA; Department of Pharmaceutical Chemistry, College of Pharmacy, Jouf University, Sakaka 72341, Saudi Arabia.
  • Ghoneim MM; Pharmaceutical Organic Chemistry Department, Faculty of Pharmacy, Beni-Suef University, Beni-Suef 62514, Egypt.
  • Shaker ME; Department of Pharmacy Practice, College of Pharmacy, AlMaarefa University, Ad Diriyah 13713, Saudi Arabia.
  • El-Sherbiny M; Pharmacognosy and Medicinal Plants Department, Faculty of Pharmacy, Al-Azhar University, Cairo 11884, Egypt.
  • Almohaimeed HM; Department of Pharmacology, College of Pharmacy, Jouf University, Sakaka 72341, Saudi Arabia.
  • Gahtori P; Department of Pharmacology & Toxicology, Faculty of Pharmacy, Mansoura University, Mansoura 35516, Egypt.
  • Kim H; Department of Basic Medical Sciences, College of Medicine, AlMaarefa University, Riyadh 11597, Saudi Arabia.
  • Mathew B; Department of Anatomy, Faculty of Medicine, Mansoura University, Mansoura 35516, Egypt.
Molecules ; 28(16)2023 Aug 21.
Article em En | MEDLINE | ID: mdl-37630420

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Doença de Parkinson / Antipsicóticos / Isatina / Neuroblastoma Limite: Humans Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Doença de Parkinson / Antipsicóticos / Isatina / Neuroblastoma Limite: Humans Idioma: En Ano de publicação: 2023 Tipo de documento: Article