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5-HT6 receptor antagonists. Design, synthesis, and structure-activity relationship of substituted 2-(1-methyl-4-piperazinyl)pyridines.
Galezowski, Michal; Fabritius, Charles-Henry; Pesonen, Ullamari; Salo, Harri; Olszak-Plachta, Marta; Czerwinska, Klaudia; Adamczyk, Justyna; Król, Marcin; Prusis, Peteris; Sieprawska-Lupa, Magdalena; Mikulski, Maciej; Kuokkanen, Katja; Obuchowicz, Radoslaw; Korjamo, Timo; Jalava, Niina; Nikiforuk, Agnieszka; Nowak, Mateusz.
Afiliação
  • Galezowski M; Ryvu Therapeutics S.A., Sternbacha Street 2, 30-394 Kraków, Poland. Electronic address: michal.galezowski@ryvu.com.
  • Fabritius CH; Ryvu Therapeutics S.A., Sternbacha Street 2, 30-394 Kraków, Poland.
  • Pesonen U; Orion Corporation, Orion Pharma, Orionintie 1A, 02200 Espoo, Finland.
  • Salo H; Orion Corporation, Orion Pharma, Orionintie 1A, 02200 Espoo, Finland.
  • Olszak-Plachta M; Ryvu Therapeutics S.A., Sternbacha Street 2, 30-394 Kraków, Poland.
  • Czerwinska K; Ryvu Therapeutics S.A., Sternbacha Street 2, 30-394 Kraków, Poland.
  • Adamczyk J; Ryvu Therapeutics S.A., Sternbacha Street 2, 30-394 Kraków, Poland.
  • Król M; Ryvu Therapeutics S.A., Sternbacha Street 2, 30-394 Kraków, Poland.
  • Prusis P; Orion Corporation, Orion Pharma, Orionintie 1A, 02200 Espoo, Finland.
  • Sieprawska-Lupa M; Ryvu Therapeutics S.A., Sternbacha Street 2, 30-394 Kraków, Poland.
  • Mikulski M; Ryvu Therapeutics S.A., Sternbacha Street 2, 30-394 Kraków, Poland.
  • Kuokkanen K; Orion Corporation, Orion Pharma, Orionintie 1A, 02200 Espoo, Finland.
  • Obuchowicz R; Ryvu Therapeutics S.A., Sternbacha Street 2, 30-394 Kraków, Poland.
  • Korjamo T; Orion Corporation, Orion Pharma, Orionintie 1A, 02200 Espoo, Finland.
  • Jalava N; Orion Corporation, Orion Pharma, Orionintie 1A, 02200 Espoo, Finland.
  • Nikiforuk A; Department of Behavioral Neuroscience and Drug Development, Maj Institute of Pharmacology Polish Academy of Sciences, 12 Smetna Street, 31-343 Kraków, Poland.
  • Nowak M; Ryvu Therapeutics S.A., Sternbacha Street 2, 30-394 Kraków, Poland.
Bioorg Med Chem Lett ; 96: 129497, 2023 11 15.
Article em En | MEDLINE | ID: mdl-37806499

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Piridinas / Antagonistas da Serotonina Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Piridinas / Antagonistas da Serotonina Idioma: En Ano de publicação: 2023 Tipo de documento: Article