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Multitargeted inhibition of key enzymes associated with diabetes and Alzheimer's disease by 1,3,4-oxadiazole derivatives: Synthesis, in vitro screening, and computational studies.
Fatima, Bibi; Saleem, Faiza; Salar, Uzma; Chigurupati, Sridevi; Felemban, Shatha G; Ul-Haq, Zaheer; Tariq, Syeda S; Almahmoud, Suliman A; Taha, Muhammad; Shah, Syed T A; Khan, Khalid M.
Afiliação
  • Fatima B; H. E. J. Research Institute of Chemistry, International Center for Chemical and Biological Sciences, University of Karachi, Karachi, Pakistan.
  • Saleem F; H. E. J. Research Institute of Chemistry, International Center for Chemical and Biological Sciences, University of Karachi, Karachi, Pakistan.
  • Salar U; Dr. Panjwani Center for Molecular Medicine and Drug Research, International Center for Chemical and Biological Sciences, University of Karachi, Karachi, Pakistan.
  • Chigurupati S; Department of Medicinal Chemistry and Pharmacognosy, College of Pharmacy, Qassim University, Buraidah, Saudi Arabia.
  • Felemban SG; Department of Medical Laboratory Science, Fakeeh College for Medical Sciences, Jeddah, Saudi Arabia.
  • Ul-Haq Z; Dr. Panjwani Center for Molecular Medicine and Drug Research, International Center for Chemical and Biological Sciences, University of Karachi, Karachi, Pakistan.
  • Tariq SS; Dr. Panjwani Center for Molecular Medicine and Drug Research, International Center for Chemical and Biological Sciences, University of Karachi, Karachi, Pakistan.
  • Almahmoud SA; Department of Medicinal Chemistry and Pharmacognosy, College of Pharmacy, Qassim University, Buraidah, Saudi Arabia.
  • Taha M; Department of Clinical Pharmacy, Institute for Research and Medical Consultations (IRMC), Imam Abdulrahman Bin Faisal University, Dammam, Saudi Arabia.
  • Shah STA; Department of Education, Sukkur IBA University, Sukkur, Pakistan.
  • Khan KM; H. E. J. Research Institute of Chemistry, International Center for Chemical and Biological Sciences, University of Karachi, Karachi, Pakistan.
Arch Pharm (Weinheim) ; 356(12): e2300384, 2023 Dec.
Article em En | MEDLINE | ID: mdl-37806747

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Diabetes Mellitus / Doença de Alzheimer Tipo de estudo: Diagnostic_studies / Risk_factors_studies / Screening_studies Limite: Humans Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Diabetes Mellitus / Doença de Alzheimer Tipo de estudo: Diagnostic_studies / Risk_factors_studies / Screening_studies Limite: Humans Idioma: En Ano de publicação: 2023 Tipo de documento: Article