Detalhe da pesquisa
1.
Mono- and multimeric PSMA-targeting small molecule-thorium-227 conjugates for optimized efficacy and biodistribution in preclinical models.
Eur J Nucl Med Mol Imaging
; 51(3): 669-680, 2024 Feb.
Artigo
em Inglês
| MEDLINE | ID: mdl-37882848
2.
A Novel NAMPT Inhibitor-Based Antibody-Drug Conjugate Payload Class for Cancer Therapy.
Bioconjug Chem
; 33(6): 1210-1221, 2022 06 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-35658441
3.
Discovery of potent SOS1 inhibitors that block RAS activation via disruption of the RAS-SOS1 interaction.
Proc Natl Acad Sci U S A
; 116(7): 2551-2560, 2019 02 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-30683722
4.
Discovery of Rigidified α,ß-Unsaturated Imines as New Resistance-breaking Insecticides for Malaria Vector Control.
Chimia (Aarau)
; 70(10): 694-697, 2016 Oct.
Artigo
em Inglês
| MEDLINE | ID: mdl-27779926
5.
Preclinical evaluation of BAY 1075553, a novel (18)F-labelled inhibitor of prostate-specific membrane antigen for PET imaging of prostate cancer.
Eur J Nucl Med Mol Imaging
; 41(1): 89-101, 2014 Jan.
Artigo
em Inglês
| MEDLINE | ID: mdl-23955632
6.
Changing for the Better: Discovery of the Highly Potent and Selective CDK9 Inhibitor VIP152 Suitable for Once Weekly Intravenous Dosing for the Treatment of Cancer.
J Med Chem
; 64(15): 11651-11674, 2021 08 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-34264057
7.
Radiofluorinated derivatives of 2-(phosphonomethyl)pentanedioic acid as inhibitors of prostate specific membrane antigen (PSMA) for the imaging of prostate cancer.
J Med Chem
; 55(22): 9510-20, 2012 Nov 26.
Artigo
em Inglês
| MEDLINE | ID: mdl-23025786
8.
Multiple palladium-catalyzed reactions for the synthesis of analogues of the highly potent insecticide spinosyn A.
Angew Chem Int Ed Engl
; 45(30): 5015-8, 2006 Jul 24.
Artigo
em Inglês
| MEDLINE | ID: mdl-16819747
9.
Synthesis of novel spinosyn A analogues by Pd-mediated transformations.
Chemistry
; 13(30): 8543-63, 2007.
Artigo
em Inglês
| MEDLINE | ID: mdl-17654624