Detalhe da pesquisa
1.
Potent reversible inhibition of myeloperoxidase by aromatic hydroxamates.
J Biol Chem
; 288(51): 36636-47, 2013 Dec 20.
Artigo
em Inglês
| MEDLINE | ID: mdl-24194519
2.
Ligand Discovery: High-Throughput Binding: Fluorescence Polarization (Anisotropy).
Methods Mol Biol
; 2263: 231-246, 2021.
Artigo
em Inglês
| MEDLINE | ID: mdl-33877601
3.
Discovery of 5-{4-[(7-Ethyl-6-oxo-5,6-dihydro-1,5-naphthyridin-3-yl)methyl]piperazin-1-yl}-N-methylpyridine-2-carboxamide (AZD5305): A PARP1-DNA Trapper with High Selectivity for PARP1 over PARP2 and Other PARPs.
J Med Chem
; 64(19): 14498-14512, 2021 10 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-34570508
4.
Structure-Guided Design and In-Cell Target Profiling of a Cell-Active Target Engagement Probe for PARP Inhibitors.
ACS Chem Biol
; 15(2): 325-333, 2020 02 21.
Artigo
em Inglês
| MEDLINE | ID: mdl-32017532
5.
Positioning High-Throughput CETSA in Early Drug Discovery through Screening against B-Raf and PARP1.
SLAS Discov
; 24(2): 121-132, 2019 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-30543471
6.
Discovery of AZD-2098 and AZD-1678, Two Potent and Bioavailable CCR4 Receptor Antagonists.
ACS Med Chem Lett
; 8(9): 981-986, 2017 Sep 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-28947948
7.
The discovery of MMP7 inhibitors exploiting a novel selectivity trigger.
ChemMedChem
; 6(5): 769-73, 2011 May 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-21520417
8.
An evaluation of fluorescence polarization and lifetime discriminated polarization for high throughput screening of serine/threonine kinases.
Anal Biochem
; 308(2): 223-31, 2002 Sep 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-12419333