Detalhe da pesquisa
1.
The decanoate esters of nandrolone, testosterone, and trenbolone induce steroid specific memory impairment and somatic effects in the male rat.
Horm Behav
; 161: 105501, 2024 May.
Artigo
em Inglês
| MEDLINE | ID: mdl-38368844
2.
The Discovery of New Inhibitors of Insulin-Regulated Aminopeptidase by a High-Throughput Screening of 400,000 Drug-like Compounds.
Int J Mol Sci
; 25(7)2024 Apr 06.
Artigo
em Inglês
| MEDLINE | ID: mdl-38612894
3.
Inhibition of Insulin-Regulated Aminopeptidase by Imidazo [1,5-α]pyridines-Synthesis and Evaluation.
Int J Mol Sci
; 25(5)2024 Feb 21.
Artigo
em Inglês
| MEDLINE | ID: mdl-38473764
4.
Two-Chamber Aminocarbonylation of Aryl Bromides and Triflates Using Amino Acids as Nucleophiles.
J Org Chem
; 88(18): 12978-12985, 2023 Sep 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-37639573
5.
Hydrogen Peroxide Induced Toxicity Is Reversed by the Macrocyclic IRAP-Inhibitor HA08 in Primary Hippocampal Cell Cultures.
Curr Issues Mol Biol
; 44(10): 5000-5012, 2022 Oct 18.
Artigo
em Inglês
| MEDLINE | ID: mdl-36286055
6.
Angiotensin II AT2 receptor ligands with phenylthiazole scaffolds.
Bioorg Med Chem
; 65: 116790, 2022 07 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-35550979
7.
2-Alkyl substituted benzimidazoles as a new class of selective AT2 receptor ligands.
Bioorg Med Chem
; 66: 116804, 2022 07 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-35576659
8.
N-(Methyloxycarbonyl)thiophene sulfonamides as high affinity AT2 receptor ligands.
Bioorg Med Chem
; 29: 115859, 2021 01 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-33309749
9.
Regio- and Stereoselective Synthesis of Allylic Spiroethers (Spirobenzofuranes) via an Intramolecular Mizoroki-Heck Reaction.
J Org Chem
; 85(12): 7648-7657, 2020 06 19.
Artigo
em Inglês
| MEDLINE | ID: mdl-32083867
10.
Trastuzumab cotreatment improves survival of mice with PC-3 prostate cancer xenografts treated with the GRPR antagonist 177 Lu-DOTAGA-PEG2 -RM26.
Int J Cancer
; 145(12): 3347-3358, 2019 12 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-31077356
11.
A convenient transesterification method for synthesis of AT2 receptor ligands with improved stability in human liver microsomes.
Bioorg Med Chem Lett
; 28(3): 519-522, 2018 02 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-29279275
12.
Palladium(0)-Catalyzed Carbonylative One-Pot Synthesis of N-Acylguanidines.
J Org Chem
; 82(23): 12520-12529, 2017 12 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-29027801
13.
Synthesis and in vitro evaluation of 5-substituted benzovesamicol analogs containing N-substituted amides as potential positron emission tomography tracers for the vesicular acetylcholine transporter.
Bioorg Med Chem
; 25(19): 5095-5106, 2017 10 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-28185725
14.
Synthesis of 11C-Labelled Ureas by Palladium(II)-Mediated Oxidative Carbonylation.
Molecules
; 22(10)2017 Oct 10.
Artigo
em Inglês
| MEDLINE | ID: mdl-28994734
15.
Binding to and Inhibition of Insulin-Regulated Aminopeptidase by Macrocyclic Disulfides Enhances Spine Density.
Mol Pharmacol
; 89(4): 413-24, 2016 Apr.
Artigo
em Inglês
| MEDLINE | ID: mdl-26769413
16.
Rapid and Efficient Conversion of (11) CO2 to (11) CO through Silacarboxylic Acids: Applications in Pd-Mediated Carbonylations.
Chemistry
; 21(49): 17601-4, 2015 Dec 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-26492852
17.
Synthesis of 4-quinolones via a carbonylative Sonogashira cross-coupling using molybdenum hexacarbonyl as a CO source.
J Org Chem
; 80(3): 1464-71, 2015 Feb 06.
Artigo
em Inglês
| MEDLINE | ID: mdl-25575042
18.
N-Substituted pyrazole-3-carboxamides as inhibitors of human 15-lipoxygenase.
Bioorg Med Chem Lett
; 25(15): 3017-23, 2015 Aug 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-26037319
19.
3-Substituted pyrazoles and 4-substituted triazoles as inhibitors of human 15-lipoxygenase-1.
Bioorg Med Chem Lett
; 25(15): 3024-9, 2015 Aug 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-26037322
20.
Virtual Screening for Transition State Analogue Inhibitors of IRAP Based on Quantum Mechanically Derived Reaction Coordinates.
J Chem Inf Model
; 55(9): 1984-93, 2015 Sep 28.
Artigo
em Inglês
| MEDLINE | ID: mdl-26252078