Detalhe da pesquisa
1.
Structural and conformational determinants of macrocycle cell permeability.
Nat Chem Biol
; 12(12): 1065-1074, 2016 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-27748751
2.
Erratum: Structural and conformational determinants of macrocycle cell permeability.
Nat Chem Biol
; 13(8): 922, 2017 Jul 18.
Artigo
em Inglês
| MEDLINE | ID: mdl-28853740
3.
Synthesis of stereochemically and skeletally diverse fused ring systems from functionalized C-glycosides.
J Org Chem
; 78(11): 5160-71, 2013 Jun 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-23692141
4.
Synthesis and profiling of a diverse collection of azetidine-based scaffolds for the development of CNS-focused lead-like libraries.
J Org Chem
; 77(17): 7187-211, 2012 Sep 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-22853001
5.
Large-scale synthesis of all stereoisomers of a 2,3-unsaturated C-glycoside scaffold.
J Org Chem
; 76(6): 1898-901, 2011 Mar 18.
Artigo
em Inglês
| MEDLINE | ID: mdl-21341742
6.
An aldol-based build/couple/pair strategy for the synthesis of medium- and large-sized rings: discovery of macrocyclic histone deacetylase inhibitors.
J Am Chem Soc
; 132(47): 16962-76, 2010 Dec 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-21067169
7.
Identification of Highly Specific Diversity-Oriented Synthesis-Derived Inhibitors of Clostridium difficile.
ACS Infect Dis
; 3(5): 349-359, 2017 05 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-28215073
8.
Novel diversity-oriented synthesis-derived respiratory syncytial virus inhibitors identified via a high throughput replicon-based screen.
Antiviral Res
; 131: 19-25, 2016 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-27059228
9.
Impact of stereospecific intramolecular hydrogen bonding on cell permeability and physicochemical properties.
J Med Chem
; 57(6): 2746-54, 2014 Mar 27.
Artigo
em Inglês
| MEDLINE | ID: mdl-24524242
10.
Practical, scalable, high-throughput approaches to eta3-pyranyl and eta3-pyridinyl organometallic enantiomeric scaffolds using the Achmatowicz reaction.
J Org Chem
; 73(3): 882-8, 2008 Feb 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-18171075