Detalhe da pesquisa
1.
Synthesis of [15 N]-cholamine bromide hydrobromide.
J Labelled Comp Radiopharm
; 61(4): 391-394, 2018 04.
Artigo
em Inglês
| MEDLINE | ID: mdl-29278650
2.
Scaffold hopping towards potent and selective JAK3 inhibitors: discovery of novel C-5 substituted pyrrolopyrazines.
Bioorg Med Chem Lett
; 24(21): 4969-75, 2014 Nov 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-25262541
3.
Exploration of a new series of CCR5 antagonists: multi-dimensional optimization of a sub-series containing N-substituted pyrazoles.
Bioorg Med Chem Lett
; 20(16): 4753-6, 2010 Aug 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-20643548
4.
Evaluation of amide replacements in CCR5 antagonists as a means to increase intrinsic permeability. Part 2: SAR optimization and pharmacokinetic profile of a homologous azacyle series.
Bioorg Med Chem Lett
; 20(22): 6802-7, 2010 Nov 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-20855212
5.
Evaluation of a 3-amino-8-azabicyclo[3.2.1]octane replacement in the CCR5 antagonist maraviroc.
Bioorg Med Chem Lett
; 20(5): 1674-6, 2010 Mar 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-20137937
6.
Evaluation of secondary amide replacements in a series of CCR5 antagonists as a means to increase intrinsic membrane permeability. Part 1: Optimization of gem-disubstituted azacycles.
Bioorg Med Chem Lett
; 20(2): 704-8, 2010 Jan 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-20004099
7.
Evaluation of a 4-aminopiperidine replacement in several series of CCR5 antagonists.
Bioorg Med Chem Lett
; 20(6): 1830-3, 2010 Mar 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-20176481
8.
Novel hexahydropyrrolo[3,4-c]pyrrole CCR5 antagonists.
Bioorg Med Chem Lett
; 20(10): 3116-9, 2010 May 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-20417098
9.
Discovery of N-[4-[6-tert-butyl-5-methoxy-8-(6-methoxy-2-oxo-1H-pyridin-3-yl)-3-quinolyl]phenyl]methanesulfonamide (RG7109), a potent inhibitor of the hepatitis C virus NS5B polymerase.
J Med Chem
; 57(5): 1914-31, 2014 Mar 13.
Artigo
em Inglês
| MEDLINE | ID: mdl-24195700
10.
Small molecule antagonists of the chemokine receptor CCR5.
Curr Top Med Chem
; 10(13): 1299-338, 2010.
Artigo
em Inglês
| MEDLINE | ID: mdl-20536424
11.
Synthesis of base-modified dihydropacidamycins.
Bioorg Med Chem Lett
; 12(7): 1121-3, 2002 Apr 08.
Artigo
em Inglês
| MEDLINE | ID: mdl-11909731
12.
Synthetic dihydropacidamycin antibiotics: a modified spectrum of activity for the pacidamycin class.
Bioorg Med Chem Lett
; 13(19): 3305-9, 2003 Oct 06.
Artigo
em Inglês
| MEDLINE | ID: mdl-12951115
13.
Quinazolinone-based fungal efflux pump inhibitors. Part 1: Discovery of an (N-methylpiperazine)-containing derivative with activity in clinically relevant Candida spp.
Bioorg Med Chem Lett
; 14(20): 5127-31, 2004 Oct 18.
Artigo
em Inglês
| MEDLINE | ID: mdl-15380213
14.
Quinazolinone fungal efflux pump inhibitors. Part 2: In vitro structure-activity relationships of (N-methyl-piperazinyl)-containing derivatives.
Bioorg Med Chem Lett
; 14(20): 5133-7, 2004 Oct 18.
Artigo
em Inglês
| MEDLINE | ID: mdl-15380214