Detalhe da pesquisa
1.
Isopropyl quinoxaline-7-carboxylate 1,4-di-N-oxide derivatives induce regulated necrosis-like cell death on Leishmania (Leishmania) mexicana.
Parasitol Res
; 117(1): 45-58, 2018 Jan.
Artigo
em Inglês
| MEDLINE | ID: mdl-29159705
2.
Anti-Mycobacterium tuberculosis Activity of Esters of Quinoxaline 1,4-Di-N-Oxide.
Molecules
; 23(6)2018 06 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-29914062
3.
Trypanocidal Activity of Quinoxaline 1,4 Di-N-oxide Derivatives as Trypanothione Reductase Inhibitors.
Molecules
; 22(2)2017 Feb 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-28157150
4.
Anti-Trypanosoma cruzi and anti-leishmanial activity by quinoxaline-7-carboxylate 1,4-di-N-oxide derivatives.
Parasitol Res
; 113(6): 2027-35, 2014 Jun.
Artigo
em Inglês
| MEDLINE | ID: mdl-24691716
5.
Synthesis, biological evaluation and structure-activity relationships of new quinoxaline derivatives as anti-Plasmodium falciparum agents.
Molecules
; 19(2): 2166-80, 2014 Feb 18.
Artigo
em Inglês
| MEDLINE | ID: mdl-24552985
6.
Synthesis and in vitro evaluation of new ethyl and methyl quinoxaline-7-carboxylate 1,4-di-N-oxide against Entamoeba histolytica.
Bioorg Med Chem
; 21(15): 4550-8, 2013 Aug 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-23787289
7.
New amide derivatives of quinoxaline 1,4-di-N-oxide with leishmanicidal and antiplasmodial activities.
Molecules
; 18(4): 4718-27, 2013 Apr 22.
Artigo
em Inglês
| MEDLINE | ID: mdl-23609622
8.
New quinoxaline derivatives as potential MT1 and MT2 receptor ligands.
Molecules
; 17(7): 7737-57, 2012 Jun 25.
Artigo
em Inglês
| MEDLINE | ID: mdl-22732886
9.
Antiplasmodial and leishmanicidal activities of 2-cyano-3-(4-phenylpiperazine-1-carboxamido) quinoxaline 1,4-dioxide derivatives.
Molecules
; 17(8): 9451-61, 2012 Aug 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-22871647
10.
New 1,4-di-N-oxide-quinoxaline-2-ylmethylene isonicotinic acid hydrazide derivatives as anti-Mycobacterium tuberculosis agents.
Bioorg Med Chem Lett
; 21(12): 3699-703, 2011 Jun 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-21570839
11.
New salicylamide and sulfonamide derivatives of quinoxaline 1,4-di-N-oxide with antileishmanial and antimalarial activities.
Bioorg Med Chem Lett
; 21(15): 4498-502, 2011 Aug 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-21724395
12.
Aryl piperazine and pyrrolidine as antimalarial agents. Synthesis and investigation of structure-activity relationships.
Exp Parasitol
; 128(2): 97-103, 2011 Jun.
Artigo
em Inglês
| MEDLINE | ID: mdl-21354139
13.
Trypanocidal properties, structure-activity relationship and computational studies of quinoxaline 1,4-di-N-oxide derivatives.
Exp Parasitol
; 127(4): 745-51, 2011 Apr.
Artigo
em Inglês
| MEDLINE | ID: mdl-21272583
14.
Genetic toxicology and preliminary in vivo studies of nitric oxide donor tocopherol analogs as potential new class of antiatherogenic agents.
Drug Chem Toxicol
; 34(3): 285-93, 2011 Jul.
Artigo
em Inglês
| MEDLINE | ID: mdl-21649483
15.
Studies on log Po/w of quinoxaline di-N-oxides: a comparison of RP-HPLC experimental and predictive approaches.
Molecules
; 16(9): 7893-908, 2011 Sep 13.
Artigo
em Inglês
| MEDLINE | ID: mdl-22143549
16.
Esters of quinoxaline-7-carboxylate-1,4-di-N-oxide as Trichomonas vaginalis triosephosphate isomerase inhibitors.
Acta Pharm
; 71(3): 485-495, 2021 Sep 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-36654088
17.
Anti-T. cruzi activities and QSAR studies of 3-arylquinoxaline-2-carbonitrile di-N-oxides.
Bioorg Med Chem Lett
; 20(16): 4831-5, 2010 Aug 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-20634064
18.
DNA strand cleaving properties and hypoxia-selective cytotoxicity of 7-chloro-2-thienylcarbonyl-3-trifluoromethylquinoxaline 1,4-dioxide.
Bioorg Med Chem
; 18(9): 3125-32, 2010 May 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-20371184
19.
New 3-methylquinoxaline-2-carboxamide 1,4-di-N-oxide derivatives as anti-Mycobacterium tuberculosis agents.
Bioorg Med Chem
; 18(7): 2713-9, 2010 Apr 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-20233660
20.
Building a MCHR1 homology model provides insight into the receptor-antagonist contacts that are important for the development of new anti-obesity agents.
Bioorg Med Chem
; 18(21): 7365-79, 2010 Nov 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-20932767