Detalhe da pesquisa
1.
Discovery of 5-(2-chloro-4'-(1H-imidazol-1-yl)-[1,1'-biphenyl]-4-yl)-1H-tetrazole as potent and orally efficacious S-nitrosoglutathione reductase (GSNOR) inhibitors for the potential treatment of COPD.
Bioorg Med Chem Lett
; 28(23-24): 3766-3773, 2018 12 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-30340896
2.
Alleviating CYP and hERG liabilities by structure optimization of dihydrofuran-fused tricyclic benzo[d]imidazole series - Potent, selective and orally efficacious microsomal prostaglandin E synthase-1 (mPGES-1) inhibitors: Part-2.
Bioorg Med Chem Lett
; 28(7): 1211-1218, 2018 04 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-29519738
3.
Discovery of furan and dihydrofuran-fused tricyclic benzo[d]imidazole derivatives as potent and orally efficacious microsomal prostaglandin E synthase-1 (mPGES-1) inhibitors: Part-1.
Bioorg Med Chem Lett
; 27(23): 5131-5138, 2017 12 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-29100801
4.
Tricyclic 4,4-dimethyl-3,4-dihydrochromeno[3,4-d]imidazole derivatives as microsomal prostaglandin E2 synthase-1 (mPGES-1) inhibitors: SAR and in vivo efficacy in hyperalgesia pain model.
Bioorg Med Chem Lett
; 27(11): 2594-2601, 2017 06 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-28400234
5.
Discovery of 2-((2-chloro-6-fluorophenyl)amino)-N-(3-fluoro-5-(trifluoromethyl)phenyl)-1-methyl-7,8-dihydro-1H-[1,4]dioxino[2',3':3,4]benzo[1,2-d]imidazole-5-carboxamide as potent, selective and efficacious microsomal prostaglandin E2 synthase-1 (mPGES-1) inhibitor.
Bioorg Med Chem Lett
; 26(24): 5977-5984, 2016 12 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-27865703
6.
Synthesis of potent, substituted carbazoles as selective androgen receptor modulators (SARMs).
Bioorg Med Chem Lett
; 20(24): 7516-20, 2010 Dec 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-21036041